PDB-code
Browse kinase entries (page 97 of 282)
First 93 94 95 PreviousLast101 100 99 Next| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | DYRK1A | DYRK | CMGC | 7a52 | A | A | 3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7a52 | A | B | 3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7a53 | A | A | (3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7a53 | A | B | (3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7a55 | A | 3-(1-methylpyrazol-4-yl)-1~{h}-pyrazole-5-carboxylic acid | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7a5b | A | 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7a5d | A | A | 4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7a5d | A | B | 4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7a5l | A | A | 4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7a5l | A | B | 4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7a5n | A | 5-(2-azanylpyridin-4-yl)-~{n}-[[2,6-bis(fluoranyl)phenyl]methyl]-2-methyl-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7aj2 | A | A | 4-(4-methoxyphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7aj2 | A | B | 4-(4-methoxyphenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7aj4 | A | A | 4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7aj4 | A | B | 4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7aj5 | A | A | 4-(1-benzofuran-5-yl)pyridine-2,6-diamine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7aj5 | A | B | 4-(1-benzofuran-5-yl)pyridine-2,6-diamine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7aj7 | A | 4-(3-methylbenzimidazol-5-yl)pyridine-2,6-diamine | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7aj8 | A | A | 4-(1-benzofuran-5-yl)pyridin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7aj8 | A | B | 4-(1-benzofuran-5-yl)pyridin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7aja | A | A | 1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7aja | A | B | 1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7ajm | A | A | ~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamide | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7ajm | A | B | ~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamide | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7ajs | A | A | 4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7ajs | A | B | 4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7ajv | A | 4-(2,3-dibutylimidazo[4,5-b]pyridin-5-yl)pyridine-2,6-diamine | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7ajw | A | A | 4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7ajw | A | B | 4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7ajy | A | 4-[2-methyl-3-[(2~{r})-2-phenoxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7ak2 | A | 4-[2-methyl-3-(2-pyridin-2-yloxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7aka | A | A | 4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7aka | A | B | 4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7akb | A | A | 4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7akb | A | B | 4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7ake | A | 4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7akl | A | 4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7fhs | A | A | (5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7fhs | A | B | (5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7fht | A | A | (5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7fht | A | B | (5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7o7k | A | A | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7o7k | A | B | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7z5n | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | Show | ![]() | |
![]() | DYRK1A | DYRK | CMGC | 7zh8 | A | A | 6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 7zh8 | A | B | 6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 8c3g | A | A | n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 8c3g | A | B | n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 8c3q | A | A | rutin | Human | Show | ![]() |
![]() | DYRK1A | DYRK | CMGC | 8c3q | A | B | rutin | Human | Show | ![]() |


