Browse kinase entries (page 97 of 282)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
DYRK1ADYRKCMGC7a52AA3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-oneHumanShow
DYRK1ADYRKCMGC7a52AB3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-oneHumanShow
DYRK1ADYRKCMGC7a53AA(3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-oneHumanShow
DYRK1ADYRKCMGC7a53AB(3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-oneHumanShow
DYRK1ADYRKCMGC7a55A3-(1-methylpyrazol-4-yl)-1~{h}-pyrazole-5-carboxylic acidHumanShow
DYRK1ADYRKCMGC7a5bA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC7a5dAA4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHumanShow
DYRK1ADYRKCMGC7a5dAB4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHumanShow
DYRK1ADYRKCMGC7a5lAA4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amineHumanShow
DYRK1ADYRKCMGC7a5lAB4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amineHumanShow
DYRK1ADYRKCMGC7a5nA5-(2-azanylpyridin-4-yl)-~{n}-[[2,6-bis(fluoranyl)phenyl]methyl]-2-methyl-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHumanShow
DYRK1ADYRKCMGC7aj2AA4-(4-methoxyphenyl)pyridin-2-amineHumanShow
DYRK1ADYRKCMGC7aj2AB4-(4-methoxyphenyl)pyridin-2-amineHumanShow
DYRK1ADYRKCMGC7aj4AA4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amineHumanShow
DYRK1ADYRKCMGC7aj4AB4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amineHumanShow
DYRK1ADYRKCMGC7aj5AA4-(1-benzofuran-5-yl)pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7aj5AB4-(1-benzofuran-5-yl)pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7aj7A4-(3-methylbenzimidazol-5-yl)pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7aj8AA4-(1-benzofuran-5-yl)pyridin-2-amineHumanShow
DYRK1ADYRKCMGC7aj8AB4-(1-benzofuran-5-yl)pyridin-2-amineHumanShow
DYRK1ADYRKCMGC7ajaAA1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazineHumanShow
DYRK1ADYRKCMGC7ajaAB1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazineHumanShow
DYRK1ADYRKCMGC7ajmAA~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamideHumanShow
DYRK1ADYRKCMGC7ajmAB~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamideHumanShow
DYRK1ADYRKCMGC7ajsAA4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7ajsAB4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7ajvA4-(2,3-dibutylimidazo[4,5-b]pyridin-5-yl)pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7ajwAA4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7ajwAB4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7ajyA4-[2-methyl-3-[(2~{r})-2-phenoxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7ak2A4-[2-methyl-3-(2-pyridin-2-yloxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7akaAA4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7akaAB4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7akbAA4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7akbAB4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7akeA4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7aklA4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamineHumanShow
DYRK1ADYRKCMGC7fhsAA(5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHumanShow
DYRK1ADYRKCMGC7fhsAB(5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHumanShow
DYRK1ADYRKCMGC7fhtAA(5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHumanShow
DYRK1ADYRKCMGC7fhtAB(5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHumanShow
DYRK1ADYRKCMGC7o7kAAn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC7o7kABn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC7z5nA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHumanShow
DYRK1ADYRKCMGC7zh8AA6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridineHumanShow
DYRK1ADYRKCMGC7zh8AB6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridineHumanShow
DYRK1ADYRKCMGC8c3gAAn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC8c3gABn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHumanShow
DYRK1ADYRKCMGC8c3qAArutinHumanShow
DYRK1ADYRKCMGC8c3qABrutinHumanShow
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