PDB-code
Search results (10 entries covering 2 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | JAK1 | JakA | TK | 4e4l | D | B | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | Show | ![]() |
![]() | JAK1 | JakA | TK | 4e4l | A | A | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | Show | ![]() |
![]() | JAK2 | JakA | TK | 4e4m | A | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | Show | ![]() | |
![]() | JAK1 | JakA | TK | 4e4l | D | A | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | Show | ![]() |
![]() | JAK1 | JakA | TK | 4e4l | B | B | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | Show | ![]() |
![]() | JAK2 | JakA | TK | 4e4m | D | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | Show | ![]() | |
![]() | JAK2 | JakA | TK | 4e4m | B | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | Show | ![]() | |
![]() | JAK2 | JakA | TK | 4e4m | E | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | Show | ![]() | |
![]() | JAK1 | JakA | TK | 4e4l | B | A | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | Show | ![]() |
![]() | JAK1 | JakA | TK | 4e4l | A | B | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | Show | ![]() |


