PDB-code
Search results (10 entries covering 4 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | HASPIN (Haspin) | Haspin | Other | 4qtc | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |
![]() | MAPK8 (JNK1) | MAPK | CMGC | 4qtd | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |
![]() | MAPK8 (JNK1) | MAPK | CMGC | 4qtd | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |
![]() | MAPK3 (Erk1) | MAPK | CMGC | 4qtb | B | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |
![]() | MAPK3 (Erk1) | MAPK | CMGC | 4qtb | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qta | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |
![]() | MAPK1 (Erk2) | MAPK | CMGC | 4qta | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |
![]() | MAPK3 (Erk1) | MAPK | CMGC | 4qtb | B | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |
![]() | MAPK3 (Erk1) | MAPK | CMGC | 4qtb | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |
![]() | HASPIN (Haspin) | Haspin | Other | 4qtc | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | Show | ![]() |


