 
		
	                PDB-code
	                
	                        
	                
	        
		Search results (10 entries covering 4 PDB structures)
 
				| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File | 
|---|---|---|---|---|---|---|---|---|---|---|
|  | JAK2-b | JakB | TK | 6brw | A | A | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show |  | 
|  | STK4 (MST1) | STE20 | STE | 8a5j | A | B | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show |  | 
|  | STK4 (MST1) | STE20 | STE | 8a5j | A | A | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show |  | 
|  | STK3 (MST2) | STE20 | STE | 8a66 | A | A | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show |  | 
|  | STK3 (MST2) | STE20 | STE | 8a66 | A | B | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show |  | 
|  | STK3 (MST2) | STE20 | STE | 5dh3 | B | B | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show |  | 
|  | JAK2-b | JakB | TK | 6brw | A | B | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show |  | 
|  | STK3 (MST2) | STE20 | STE | 5dh3 | A | A | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show |  | 
|  | STK3 (MST2) | STE20 | STE | 5dh3 | B | A | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show |  | 
|  | STK3 (MST2) | STE20 | STE | 5dh3 | A | B | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | Show |  | 
