Search results (6 entries covering 3 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
EGFREGFRTK8a2bAB(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHumanShow
EGFREGFRTK8a2aAB(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHumanShow
EGFREGFRTK8a27AA(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHumanShow
EGFREGFRTK8a2aAA(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHumanShow
EGFREGFRTK8a27AB(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHumanShow
EGFREGFRTK8a2bAA(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHumanShow