Search results (36 entries covering 17 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
PI4KBPIKAtypical4d0mgn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical8vofAmethyl 2-chloro-5-(methyl{(8r)-3-[4-(methylcarbamoyl)phenyl]pyrazolo[1,5-a]pyridine-5-carbonyl}amino)benzoateHumanShow
PI4KBPIKAtypical4d0mCn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical4d0mIn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical4d0mYn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical5fblA~{n}-[2-[[6-chloranyl-3-(4-methoxy-3-morpholin-4-ylsulfonyl-phenyl)-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHumanShow
PI4KBPIKAtypical5fbwA~{n}-[2-[[6-chloranyl-3-[4-methoxy-3-[[(2~{r})-1-oxidanylbutan-2-yl]sulfamoyl]phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHumanShow
PI4KBPIKAtypical4d0mMn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical4d0mcn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical4d0mQn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical8q6fAC3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidineHumanShow
PI4KBPIKAtypical5fbqA~{n}-[2-[[6-chloranyl-3-[3-[4-(hydroxymethyl)piperidin-1-yl]sulfonyl-4-methoxy-phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHumanShow
PI4KBPIKAtypical4d0lEn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical4d0mWn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical4d0lAn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical4d0mSn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical6gl3A(3~{s})-4-(6-azanyl-1-methyl-pyrazolo[3,4-d]pyrimidin-4-yl)-~{n}-(4-methoxy-2-methyl-phenyl)-3-methyl-piperazine-1-carboxamideHumanShow
PI4KBPIKAtypical5euqE~{n}-[5-[3-[[(4-hydroxyphenyl)amino]-bis(oxidanyl)-$l^{4}-sulfanyl]-4-methoxy-phenyl]-4-methyl-1,3-thiazol-2-yl]cyclopentanecarboxamideHumanShow
PI4KBPIKAtypical4waeAadenosine-5'-triphosphateHumanShow
PI4KBPIKAtypical4d0mAn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical8q6gAC3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHumanShow
PI4KBPIKAtypical5c46E-HumanShow
PI4KBPIKAtypical4d0mOn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical5c4gEn~2~-[7-(3,4-dimethoxyphenyl)quinoxalin-2-yl]-n-methylglycinamideHumanShow
PI4KBPIKAtypical5fbvA~{n}-[2-[[6-chloranyl-3-[3-(2-hydroxyethylsulfamoyl)-4-methoxy-phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHumanShow
PI4KBPIKAtypical4d0lCn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical8q6fAA3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidineHumanShow
PI4KBPIKAtypical8q6gAA3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHumanShow
PI4KBPIKAtypical8q6hAA3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHumanShow
PI4KBPIKAtypical5fbrA~{n}-[2-[[3-[3-[(4-azanylcyclohexyl)sulfamoyl]-4-methoxy-phenyl]-6-chloranyl-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHumanShow
PI4KBPIKAtypical4wagA6-chloro-3-(3,4-dimethoxyphenyl)-2-methylimidazo[1,2-b]pyridazin-8-amineHumanShow
PI4KBPIKAtypical8q6fAB3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidineHumanShow
PI4KBPIKAtypical4d0mGn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHumanShow
PI4KBPIKAtypical6gl3B-HumanShow
PI4KBPIKAtypical8q6gAB3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHumanShow
PI4KBPIKAtypical8q6hAB3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHumanShow