Search results (24 entries covering 15 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
TTBK1TTBKCK14nfnAB3-({5-[(4-amino-4-methylpiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-bromophenolHumanShow
TTBK1TTBKCK14nfnAA3-({5-[(4-amino-4-methylpiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-bromophenolHumanShow
TTBK1TTBKCK17zhpAB1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-ethyl-pent-1-yn-3-olHumanShow
TTBK1TTBKCK17qhwA~{n}-[4-(4-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHumanShow
TTBK1TTBKCK18xpzA-HumanShow
TTBK1TTBKCK17jxxAA4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHumanShow
TTBK1TTBKCK17zhoAB4-[3-(2-azanylpyrimidin-4-yl)-1~{h}-indol-5-yl]-2-methyl-but-3-yn-2-olHumanShow
TTBK1TTBKCK14btmBmethyl 2-bromo-5-(7h-pyrrolo[2,3-d]pyrimidin-4-ylamino)benzoateHumanShow
TTBK1TTBKCK17zhqAA(3~{s})-1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-methyl-pent-1-yn-3-olHumanShow
TTBK1TTBKCK14btmAmethyl 2-bromo-5-(7h-pyrrolo[2,3-d]pyrimidin-4-ylamino)benzoateHumanShow
TTBK1TTBKCK17jxyA(3s)-1-[1-(2-aminopyrimidin-4-yl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-methylpent-1-yn-3-olHumanShow
TTBK1TTBKCK17zhnAB4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHumanShow
TTBK1TTBKCK17zhoAA4-[3-(2-azanylpyrimidin-4-yl)-1~{h}-indol-5-yl]-2-methyl-but-3-yn-2-olHumanShow
TTBK1TTBKCK14btjAadenosine-5'-diphosphateHumanShow
TTBK1TTBKCK17zhqAB(3~{s})-1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-methyl-pent-1-yn-3-olHumanShow
TTBK1TTBKCK14btjBadenosine-5'-triphosphateHumanShow
TTBK1TTBKCK17q8wAA~{n}-(4-methoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHumanShow
TTBK1TTBKCK14nfmA-HumanShow
TTBK1TTBKCK17q8wAB~{n}-(4-methoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHumanShow
TTBK1TTBKCK14btkA4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHumanShow
TTBK1TTBKCK17zhpAA1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-ethyl-pent-1-yn-3-olHumanShow
TTBK1TTBKCK17zhnAA4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHumanShow
TTBK1TTBKCK17q8vA~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHumanShow
TTBK1TTBKCK17jxxAB4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHumanShow