Search results (9 entries covering 4 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
VRK2VRKCK12v62BB-HumanShow
VRK2VRKCK15uu1A(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHumanShow
VRK2VRKCK12v62AB-HumanShow
VRK2VRKCK16ncgB4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamideHumanShow
VRK2VRKCK12v62BA-HumanShow
VRK2VRKCK18q1zAA2-[4-[[4-[(3-~{tert}-butyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]ethanenitrileHumanShow
VRK2VRKCK12v62AA-HumanShow
VRK2VRKCK16ncgA4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamideHumanShow
VRK2VRKCK18q1zAB2-[4-[[4-[(3-~{tert}-butyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]ethanenitrileHumanShow