Search results (19 entries covering 10 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK5CDKCMGC4au8AB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHumanShow
CDK5CDKCMGC1h4lA-HumanShow
CDK5CDKCMGC7vdrA(1r)-1-[7-[(2-fluoranyl-4-pyrazol-1-yl-phenyl)amino]-1,6-naphthyridin-2-yl]-1-(1-methylpiperidin-4-yl)ethanolHumanShow
CDK5CDKCMGC4au8BB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHumanShow
CDK5CDKCMGC7vdpA[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHumanShow
CDK5CDKCMGC1unlAr-roscovitineHumanShow
CDK5CDKCMGC1unlB-HumanShow
CDK5CDKCMGC7vdqA2-[[7-[[2-fluoranyl-4-[3-(hydroxymethyl)pyrazol-1-yl]phenyl]amino]-1,6-naphthyridin-2-yl]-(1-methylpiperidin-4-yl)amino]ethanoic acidHumanShow
CDK5CDKCMGC7vdsAA5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHumanShow
CDK5CDKCMGC1unhA(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHumanShow
CDK5CDKCMGC3o0gA-HumanShow
CDK5CDKCMGC1unhB(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHumanShow
CDK5CDKCMGC3o0gB{4-amino-2-[(4-chlorophenyl)amino]-1,3-thiazol-5-yl}(3-nitrophenyl)methanoneHumanShow
CDK5CDKCMGC7vdsAB5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHumanShow
CDK5CDKCMGC1ungB6-phenyl[5h]pyrrolo[2,3-b]pyrazineHumanShow
CDK5CDKCMGC1ungA6-phenyl[5h]pyrrolo[2,3-b]pyrazineHumanShow
CDK5CDKCMGC1h4lB-HumanShow
CDK5CDKCMGC4au8AA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHumanShow
CDK5CDKCMGC4au8BA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHumanShow