Search results (18 entries covering 11 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
CDK7CDKCMGC6o9l8-HumanShow
CDK7CDKCMGC8p4zAA2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amineHumanShow
CDK7CDKCMGC8p4zAB2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amineHumanShow
CDK7CDKCMGC8pyrAB-HumanShow
CDK7CDKCMGC6xd3Jn-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)-4-{[4-(dimethylamino)butanoyl]amino}benzamideHumanShow
CDK7CDKCMGC1ua2Cadenosine-5'-triphosphateHumanShow
CDK7CDKCMGC7b5oJA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHumanShow
CDK7CDKCMGC7nvr8-HumanShow
CDK7CDKCMGC7b5qJA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHumanShow
CDK7CDKCMGC7b5oJB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHumanShow
CDK7CDKCMGC1ua2Dadenosine-5'-triphosphateHumanShow
CDK7CDKCMGC7b5qJB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHumanShow
CDK7CDKCMGC8byqI-HumanShow
CDK7CDKCMGC8bvwI-HumanShow
CDK7CDKCMGC6xbzJphosphothiophosphoric acid-adenylate esterHumanShow
CDK7CDKCMGC1ua2Badenosine-5'-triphosphateHumanShow
CDK7CDKCMGC1ua2Aadenosine-5'-triphosphateHumanShow
CDK7CDKCMGC8pyrAA-HumanShow