PDB-code
Search results (21 entries covering 12 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MAPK7 (Erk5) | MAPK | CMGC | 5byy | A | A | 2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 5o7i | A | A | 4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 7pus | A | B | 4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 5byz | A | A | 4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamide | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 4ic7 | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 4zsl | A | 3-amino-5-[(4-chlorophenyl)amino]-n-[(1s)-1-phenylethyl]-1h-1,2,4-triazole-1-carboxamide | Human | Show | ![]() | |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 7pus | A | A | 4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 6hkn | A | A | [2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanone | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 4ic7 | D | phosphoaminophosphonic acid-adenylate ester | Human | Show | ![]() | |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 4ic8 | B | - | Human | Show | ![]() | |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 6hkn | A | B | [2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanone | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 4ic8 | A | - | Human | Show | ![]() | |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 6hkm | A | [4-(6,7-dimethoxyquinazolin-4-yl)piperidin-1-yl]-[4-(trifluoromethyloxy)phenyl]methanone | Human | Show | ![]() | |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 4b99 | A | 11-cyclopentyl-2-[[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl-phenyl]amino]-5-methyl-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | ![]() | |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 4zsj | A | B | 3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 5byz | A | B | 4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamide | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 4zsg | A | A | 3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 5o7i | A | B | 4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamide | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 5byy | A | B | 2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 4zsg | A | B | 3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | Show | ![]() |
![]() | MAPK7 (Erk5) | MAPK | CMGC | 4zsj | A | A | 3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | Show | ![]() |


