Search results (21 entries covering 12 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
MAPK7 (Erk5)MAPKCMGC5byyAA2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHumanShow
MAPK7 (Erk5)MAPKCMGC5o7iAA4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamideHumanShow
MAPK7 (Erk5)MAPKCMGC7pusAB4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamideHumanShow
MAPK7 (Erk5)MAPKCMGC5byzAA4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamideHumanShow
MAPK7 (Erk5)MAPKCMGC4ic7Aphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK7 (Erk5)MAPKCMGC4zslA3-amino-5-[(4-chlorophenyl)amino]-n-[(1s)-1-phenylethyl]-1h-1,2,4-triazole-1-carboxamideHumanShow
MAPK7 (Erk5)MAPKCMGC7pusAA4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamideHumanShow
MAPK7 (Erk5)MAPKCMGC6hknAA[2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanoneHumanShow
MAPK7 (Erk5)MAPKCMGC4ic7Dphosphoaminophosphonic acid-adenylate esterHumanShow
MAPK7 (Erk5)MAPKCMGC4ic8B-HumanShow
MAPK7 (Erk5)MAPKCMGC6hknAB[2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanoneHumanShow
MAPK7 (Erk5)MAPKCMGC4ic8A-HumanShow
MAPK7 (Erk5)MAPKCMGC6hkmA[4-(6,7-dimethoxyquinazolin-4-yl)piperidin-1-yl]-[4-(trifluoromethyloxy)phenyl]methanoneHumanShow
MAPK7 (Erk5)MAPKCMGC4b99A11-cyclopentyl-2-[[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl-phenyl]amino]-5-methyl-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHumanShow
MAPK7 (Erk5)MAPKCMGC4zsjAB3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHumanShow
MAPK7 (Erk5)MAPKCMGC5byzAB4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamideHumanShow
MAPK7 (Erk5)MAPKCMGC4zsgAA3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHumanShow
MAPK7 (Erk5)MAPKCMGC5o7iAB4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamideHumanShow
MAPK7 (Erk5)MAPKCMGC5byyAB2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHumanShow
MAPK7 (Erk5)MAPKCMGC4zsgAB3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHumanShow
MAPK7 (Erk5)MAPKCMGC4zsjAA3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHumanShow