PDB-code
Search results (8 entries covering 4 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | PRKCA (PKCa) | PKC | AGC | 8uak | A | A | (6m)-3-amino-n-[3-(4-amino-4-methylpiperidin-1-yl)pyridin-2-yl]-6-[3-(trifluoromethyl)pyridin-2-yl]pyrazine-2-carboxamide | Human | Show | ![]() |
![]() | PRKCA (PKCa) | PKC | AGC | 4ra4 | A | (1r)-9-[(3s,4s)-1,3-dimethylpiperidin-4-yl]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | Show | ![]() | |
![]() | PRKCA (PKCa) | PKC | AGC | 3iw4 | C | 3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dione | Human | Show | ![]() | |
![]() | PRKCA (PKCa) | PKC | AGC | 8u37 | A | B | (6m)-3-amino-n-{4-[(3r,4s)-4-amino-3-methoxypiperidin-1-yl]pyridin-3-yl}-6-[3-(trifluoromethoxy)pyridin-2-yl]pyrazine-2-carboxamide | Human | Show | ![]() |
![]() | PRKCA (PKCa) | PKC | AGC | 8u37 | A | A | (6m)-3-amino-n-{4-[(3r,4s)-4-amino-3-methoxypiperidin-1-yl]pyridin-3-yl}-6-[3-(trifluoromethoxy)pyridin-2-yl]pyrazine-2-carboxamide | Human | Show | ![]() |
![]() | PRKCA (PKCa) | PKC | AGC | 3iw4 | A | 3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dione | Human | Show | ![]() | |
![]() | PRKCA (PKCa) | PKC | AGC | 3iw4 | B | 3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dione | Human | Show | ![]() | |
![]() | PRKCA (PKCa) | PKC | AGC | 8uak | A | B | (6m)-3-amino-n-[3-(4-amino-4-methylpiperidin-1-yl)pyridin-2-yl]-6-[3-(trifluoromethyl)pyridin-2-yl]pyrazine-2-carboxamide | Human | Show | ![]() |


