Search results (111 entries covering 67 PDB structures)

Your browser unfortunately does not support an HTML5 canvas. Your browser unfortunately does not support an HTML5 canvas.
#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
MAP2K1STE7STE7f2xAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE7b94Bphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE2p55A2-[(4-ethynyl-2-fluorophenyl)amino]-3,4-difluoro-n-(2-hydroxyethoxy)benzamideHumanShow
MAP2K1STE7STE7xncA~{n}-[4-[[6-(3-chloranylpyridin-4-yl)-3-methyl-1~{h}-indazol-4-yl]oxy]cyclohexyl]ethanamideHumanShow
MAP2K1STE7STE6v2wBBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE4mneEAphosphomethylphosphonic acid adenylate esterHumanShow
MAP2K1STE7STE7m0tB5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamideHumanShow
MAP2K1STE7STE4mneABphosphomethylphosphonic acid adenylate esterHumanShow
MAP2K1STE7STE7m0vBAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE4an9Aphosphomethylphosphonic acid adenylate esterHumanShow
MAP2K1STE7STE7b9lBAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE6u2gAphosphomethylphosphonic acid adenylate esterHumanShow
MAP2K1STE7STE7pqvAA8-(2-chloranyl-4-methoxy-phenyl)-7-fluoranyl-1-piperidin-4-yl-imidazo[4,5-c]quinolineHumanShow
MAP2K1STE7STE3vvhAAadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE7m0vBBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE3zm4A7-chloranyl-6-[(3s)-pyrrolidin-3-yl]oxy-2h-isoquinolin-1-oneHumanShow
MAP2K1STE7STE6pp9BAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE7b3mBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE7pqvAB8-(2-chloranyl-4-methoxy-phenyl)-7-fluoranyl-1-piperidin-4-yl-imidazo[4,5-c]quinolineHumanShow
MAP2K1STE7STE7m0yBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE6q0jCA5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHumanShow
MAP2K1STE7STE3eqgAadenosine-5'-diphosphateHumanShow
MAP2K1STE7STE7mfdBn-(3-fluoro-4-{[4-methyl-2-oxo-7-(pyrimidin-2-yloxy)-2h-chromen-3-yl]methyl}pyridin-2-yl)-n'-methylsulfuric diamideHumanShow
MAP2K1STE7STE3e8nAadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE7m0wBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE4an3Aadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE7xlpA(1~{r},3~{s})-3-[[6-[2-chloranyl-4-(4-methylpyrimidin-2-yl)oxy-phenyl]-3-methyl-1~{h}-indazol-4-yl]oxy]cyclohexan-1-amineHumanShow
MAP2K1STE7STE8chfE-HumanShow
MAP2K1STE7STE3eqcAA2-[(2-chloro-4-iodophenyl)amino]-n-{[(2r)-2,3-dihydroxypropyl]oxy}-3,4-difluorobenzamideHumanShow
MAP2K1STE7STE3dv3ABadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE6q0jCB5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHumanShow
MAP2K1STE7STE5yt3Bphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE6q0tCA5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHumanShow
MAP2K1STE7STE4arkAadenosine-5'-diphosphateHumanShow
MAP2K1STE7STE4mneHBphosphomethylphosphonic acid adenylate esterHumanShow
MAP2K1STE7STE6q0tCB5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHumanShow
MAP2K1STE7STE4u80Aphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE4u81A8-[(4-cyclopropyl-2-fluorophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-7-carboxamideHumanShow
MAP2K1STE7STE3os3Aadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE3slsBBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE3ornAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE7b9lAAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE4mneDBphosphomethylphosphonic acid adenylate esterHumanShow
MAP2K1STE7STE7umbBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE3eqbABadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE4anbA[3-(aminomethyl)-3-oxidanyl-azetidin-1-yl]-[3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]methanoneHumanShow
MAP2K1STE7STE3zlwA(1r)-1-hydroxy-1-methyl-2,3,6,7-tetrahydro-1h,5h-pyrido[3,2,1-ij]quinolin-5-oneHumanShow
MAP2K1STE7STE6v2wBAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE4mneEBphosphomethylphosphonic acid adenylate esterHumanShow
MAP2K1STE7STE3vvhCAadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE4mneAAphosphomethylphosphonic acid adenylate esterHumanShow
MAP2K1STE7STE5yt3Aphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE3eqcAB2-[(2-chloro-4-iodophenyl)amino]-n-{[(2r)-2,3-dihydroxypropyl]oxy}-3,4-difluorobenzamideHumanShow
MAP2K1STE7STE7b9lBBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE3eqbAAadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE3vvhABadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE5hzeAA(3s,4r,8s,9s,11e)-8,9,16-trihydroxy-3,4-dimethyl-14-(methylamino)-3,4,5,6,9,10-hexahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHumanShow
MAP2K1STE7STE3vvhCBadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE3dy7Aadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE3mblABadenosine-5'-diphosphateHumanShow
MAP2K1STE7STE8dgsBAphosphothiophosphoric acid-adenylate esterHumanShow
MAP2K1STE7STE8dgtBAphosphothiophosphoric acid-adenylate esterHumanShow
MAP2K1STE7STE8dgsBBphosphothiophosphoric acid-adenylate esterHumanShow
MAP2K1STE7STE8dgtBBphosphothiophosphoric acid-adenylate esterHumanShow
MAP2K1STE7STE3v04A4-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)-1h-indazole-5-carboxamideHumanShow
MAP2K1STE7STE6nybBadenosine-5'-diphosphateHumanShow
MAP2K1STE7STE6q0jDB5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHumanShow
MAP2K1STE7STE5yt3Dphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE4mneDAphosphomethylphosphonic acid adenylate esterHumanShow
MAP2K1STE7STE3slsBAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE7m0xBAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE3slsAAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE4mneHAphosphomethylphosphonic acid adenylate esterHumanShow
MAP2K1STE7STE7b7rAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE6pp9BBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE3dv3AAadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE4lmnAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE3eqfAk-252aHumanShow
MAP2K1STE7STE3wigAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE1s9jAadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE3pp1ABadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE3slsABphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE3vvhBAadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE7b7rBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE5eymAB3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHumanShow
MAP2K1STE7STE3eqdAphosphothiophosphoric acid-adenylate esterHumanShow
MAP2K1STE7STE5bx0Aethyl 2h-indazole-5-carboxylateHumanShow
MAP2K1STE7STE4u7zA5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamideHumanShow
MAP2K1STE7STE3zlyA3-amino-1h-indazole-4-carbonitrileHumanShow
MAP2K1STE7STE5hzeAB(3s,4r,8s,9s,11e)-8,9,16-trihydroxy-3,4-dimethyl-14-(methylamino)-3,4,5,6,9,10-hexahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHumanShow
MAP2K1STE7STE6q0jDA5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHumanShow
MAP2K1STE7STE3w8qAphosphothiophosphoric acid-adenylate esterHumanShow
MAP2K1STE7STE3vvhBBadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE3eqiAadenosine-5'-diphosphateHumanShow
MAP2K1STE7STE4an2AB[3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]-[3-oxidanyl-3-[(2s)-piperidin-2-yl]azetidin-1-yl]methanoneHumanShow
MAP2K1STE7STE3eqhA(2z)-bis{amino[(2-aminophenyl)sulfanyl]methylidene}butanedinitrileHumanShow
MAP2K1STE7STE3pp1AAadenosine-5'-triphosphateHumanShow
MAP2K1STE7STE7b3mAphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE3zlsA1h-pyrrolo[2,3-b]pyridine-3-carboxylic acidHumanShow
MAP2K1STE7STE4an2AA[3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]-[3-oxidanyl-3-[(2s)-piperidin-2-yl]azetidin-1-yl]methanoneHumanShow
MAP2K1STE7STE3v01An-{[(2r)-2,3-dihydroxypropyl]oxy}-3-[(2-fluoro-4-iodophenyl)amino]furo[3,2-c]pyridine-2-carboxamideHumanShow
MAP2K1STE7STE7m0zBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE5eymBA3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHumanShow
MAP2K1STE7STE3zlxA7-choro-6-[(3r)-pyrrolidin-3-ylmethoxy]isoquinolin-1(2h)-oneHumanShow
MAP2K1STE7STE7m0uB5-[(4-bromo-2-fluorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamideHumanShow
MAP2K1STE7STE5yt3Cphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE3mblAAadenosine-5'-diphosphateHumanShow
MAP2K1STE7STE7m0xBBphosphoaminophosphonic acid-adenylate esterHumanShow
MAP2K1STE7STE5eymBB3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHumanShow
MAP2K1STE7STE5eymAA3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHumanShow
MAP2K1STE7STE7b9lABphosphoaminophosphonic acid-adenylate esterHumanShow