PDB-code
Search results (10 entries covering 3 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | MAP3K8 (COT) | STE-Unique | STE | 4y85 | A | 5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amine | Human | Show | ![]() | |
![]() | MAP3K8 (COT) | STE-Unique | STE | 4y85 | C | 5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amine | Human | Show | ![]() | |
![]() | MAP3K8 (COT) | STE-Unique | STE | 5iu2 | A | A | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | Show | ![]() |
![]() | MAP3K8 (COT) | STE-Unique | STE | 4y83 | A | 5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | Show | ![]() | |
![]() | MAP3K8 (COT) | STE-Unique | STE | 4y83 | B | 5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | Show | ![]() | |
![]() | MAP3K8 (COT) | STE-Unique | STE | 5iu2 | B | B | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | Show | ![]() |
![]() | MAP3K8 (COT) | STE-Unique | STE | 5iu2 | A | B | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | Show | ![]() |
![]() | MAP3K8 (COT) | STE-Unique | STE | 4y85 | B | 5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amine | Human | Show | ![]() | |
![]() | MAP3K8 (COT) | STE-Unique | STE | 5iu2 | B | A | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | Show | ![]() |
![]() | MAP3K8 (COT) | STE-Unique | STE | 4y83 | C | 5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | Show | ![]() |


