PDB-code
Search results (31 entries covering 5 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | B | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 7mgj | A | n-methyl-4-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]pyridine-2-carboxamide | Human | Show | ![]() | |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | D | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | C | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | A | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | C | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | A | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | A | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | B | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | C | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | C | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | A | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | C | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | C | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 7mgk | A | B | n-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | D | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | D | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | A | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | D | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | B | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | B | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | C | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | D | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 7mgk | A | A | n-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yff | A | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | B | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 4yfi | B | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | B | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | D | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | A | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |
![]() | TNNI3K (HH498) | MLK | TKL | 6b5j | D | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | Show | ![]() |


