PDB-code
Search results (12 entries covering 7 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | Btk (BTK) | Tec | TK | 8s93 | A | A | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | Show |  |
| Btk (BTK) | Tec | TK | 6mny | A | A | 5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamide | Mouse | Show | |
| Btk (BTK) | Tec | TK | 8s93 | A | B | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | Show | |
| Btk (BTK) | Tec | TK | 8s9f | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | Show | | |
| Btk (BTK) | Tec | TK | 8gmb | A | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | Show | | |
| Btk (BTK) | Tec | TK | 8ff0 | A | 6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-one | Mouse | Show | | |
| Btk (BTK) | Tec | TK | 8fd9 | A | A | acalabrutinib | Mouse | Show | |
| Btk (BTK) | Tec | TK | 8fd9 | A | B | acalabrutinib | Mouse | Show | |
| Btk (BTK) | Tec | TK | 6mny | B | A | - | Mouse | Show | |
| Btk (BTK) | Tec | TK | 4xi2 | A | - | Mouse | Show | | |
| Btk (BTK) | Tec | TK | 6mny | B | B | - | Mouse | Show | |
| Btk (BTK) | Tec | TK | 6mny | A | B | 5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamide | Mouse | Show | |
