Search results (8 entries covering 6 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
RPS6KA3-b (RSK2-b)RSKbCAMK8xeyA-HumanShow
RPS6KA3-b (RSK2-b)RSKbCAMK4jg7AB(2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamideHumanShow
RPS6KA3-b (RSK2-b)RSKbCAMK4jg6A(2s)-2-cyano-3-(1h-indazol-5-yl)propanamideHumanShow
RPS6KA3-b (RSK2-b)RSKbCAMK4d9tAmethyl (2s)-3-{4-amino-7-[(1e)-3-hydroxyprop-1-en-1-yl]-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl}-2-cyanopropanoateHumanShow
RPS6KA3-b (RSK2-b)RSKbCAMK4d9uAtert-butyl (2s)-3-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl]-2-cyanopropanoateHumanShow
RPS6KA3-b (RSK2-b)RSKbCAMK4jg8AB(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHumanShow
RPS6KA3-b (RSK2-b)RSKbCAMK4jg8AA(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHumanShow
RPS6KA3-b (RSK2-b)RSKbCAMK4jg7AA(2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamideHumanShow