Mitogen-activated protein kinase kinase kinase kinase 1
Kinase structure
Kinase:MAP4K1 (HPK1)
Family:STE20
Group:STE
Species:HUMAN
IUPHAR/BPS ID:2085
PDB:6CQE
sc-PDB:
KIDFamMap:Search
Release date:2018-12-19
PubMed: 30503777
Chain:A
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 6CQE
6CQEAlternative model: AChain: A
6CQEAlternative model: AChain: B
6CQEAlternative model: BChain: B


Structural information
DFG conformation:out-like
αC-helix conformation:out
G-rich loop angle (distance):-
G-rich loop rotation:-
Quality Score:6.4
Resolution:1.89 Å
Missing Residues:4
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I3
I6
Ligand
No
No
Protein
Yes
No

Pocket alignment
Uniprot sequence:QRLGGGTYGEVFKVALKMVTLQKEILILKTCRANIVAYHGSWICMEFCGAGSLQDIYQVYLHSQKKIHRDIKGANILILADFGIS
Sequence structure:QRLG____GEVFKVALKMVTLQKEILILKTCRANIVAYHGSWICMEFCGAGSLQDIYQVYLHSQKKIHRDIKGANILILADFGIS