Mitogen-activated protein kinase 14
Kinase structure
Kinase:MAPK14 (p38a)
Family:MAPK
Group:CMGC
Species:HUMAN
IUPHAR/BPS ID:1499
PDB:6HWV
sc-PDB:
KIDFamMap:Search
Release date:2019-04-17
PubMed: 30924488
Chain:A
(Alternate) Model:A
Click to open a 3D viewer
The orthosteric binding pocket


More entries for 6HWV
6HWVAlternative model: BChain: A


Structural information
DFG conformation:out
αC-helix conformation:in
G-rich loop angle (distance):69.3° (21.1Å)
G-rich loop rotation:45.1°
Quality Score:6.4
Resolution:1.7 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I3
Ligand
No
Protein
Yes

Pocket alignment
Uniprot sequence:SPVGSGAYGSVCAVAVKKLRTYRELRLLKHMKENVIGLLDVYLVTHLMG-ADLNNIVKCYIHSADIIHRDLKPSNLAVILDFGLA
Sequence structure:SPVGSGAYGSVCAVAVKKLRTYRELRLLKHMKENVIGLLDVYLVTHLMG_ADLNNIVKCYIHSADIIHRDLKPSNLAVILDFGLA