PDB-code
Search results (360 entries covering 243 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | MAPK14 (p38a) | MAPK | CMGC | 3k3i | A | A | (3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinoline | Human | Show |  |
| MAPK14 (p38a) | MAPK | CMGC | 1bl7 | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4zth | A | B | 6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwu | A | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfi | A | A | ~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmn | A | A | 6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 4 | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv7 | A | 1-[1-(3-aminophenyl)-3-tert-butyl-1h-pyrazol-5-yl]-3-naphthalen-1-ylurea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2baj | A | 1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2,3-dichlorophenyl)urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2okr | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3obj | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsg | A | A | tak-715 | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2i0h | A | A | 2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dione | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4aac | A | n-isoxazol-3-yl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxo-quinazolin-3-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3c5u | A | 6-[4-(2-fluorophenyl)-1,3-oxazol-5-yl]-n-(1-methylethyl)-1,3-benzothiazol-2-amine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1r3c | A | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3oc1 | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3obg | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5wjj | A | A | n-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5mz3 | A | B | ~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh8 | A | B | [3-(benzyloxy)phenyl]methanol | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2fso | X | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3qud | A | A | {4-[(2-aminophenyl)amino]phenyl}(phenyl)methanone | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3bv2 | A | 5-methyl-4-[(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)amino]-n-(1-phenylethenyl)pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5b | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3ctq | A | n-benzyl-1-[5-({5-tert-butyl-2-methoxy-3-[(methylsulfonyl)amino]phenyl}carbamoyl)-2-methylphenyl]-1h-1,2,3-triazole-4-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh2 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fko | A | 3-(2-chlorophenyl)-6-(2-fluorophenoxy)-2h-indazole | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | H | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3kf7 | A | 3-{6-[2-(2,4-difluorophenyl)ethyl][1,2,4]triazolo[4,3-a]pyridin-3-yl}-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4r3c | A | A | 6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5tco | A | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulene-9-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2gfs | A | B | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3oef | X | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5a | X | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnv | A | A | 1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylurea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | A | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4dli | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2y8o | A | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6qdz | A | B | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3oef | X | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5tbe | A | ~{n}-[2,4-bis(fluoranyl)-5-[[9-(2-morpholin-4-ylethylcarbamoyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulen-3-yl]amino]phenyl]thiophene-2-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3j | A | 2-(4-fluorophenyl)-3-oxo-6-pyridin-4-yl-n-[2-(trifluoromethyl)benzyl]-2,3-dihydropyridazine-4-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | C | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hrb | A | [3-amino-2-(2-methylphenyl)-1-oxidopyridin-4-yl](2,4-difluorophenyl)methanone | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1w84 | A | 3-(2-pyridin-4-ylethyl)-1h-indole | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2gfs | A | A | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3u8w | A | 3-[3-(2-chloro-6-fluorophenyl)-5-ethyl-6-oxo-5,6-dihydro[1,2,4]triazolo[4,3-b]pyridazin-7-yl]-n-cyclopropyl-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3huc | A | A | n-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | A | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbt | A | 3-fluoro-5-morpholin-4-yl-n-[1-(2-pyridin-4-ylethyl)-1h-indol-6-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3i | A | B | (3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinoline | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnw | A | B | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3heg | A | A | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5mtx | A | B | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfo | A | B | 5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1w83 | A | n-[4-chloro-3-(pyridin-3-yloxymethyl)-phenyl]-3-fluoro- | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5mty | A | ~{n}-[2,4-bis(fluoranyl)-5-[[14-(2-hydroxyethylcarbamoyl)-2-oxidanylidene-6-tricyclo[9.4.0.0^{3,8}]pentadeca-1(15),3(8),4,6,11,13-hexaenyl]amino]phenyl]thiophene-2-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5o8v | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfb | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5etf | A | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3fsf | A | 3-(2,6-dichlorophenyl)-7-({4-[(diethylamino)methoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmk | A | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvq | A | A | n-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh9 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1bl6 | A | 4-(4-fluorophenyl)-1-cycloropropylmethyl-5-(4-pyridyl)-imidazole | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3zya | A | B | 2-amino-phenylamino-dibenzosuberone | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4ewq | A | A | 3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | B | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsi | A | B | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp2 | A | B | 1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-one | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3kq7 | A | A | n-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvq | A | B | n-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5omh | A | 1-(3-chlorophenyl)-3-methyl-4~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4ehv | A | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3mw1 | A | 8-(2,6-dichlorophenyl)-4-(2,4-difluorophenyl)-2-piperidin-4-yl-1,7-naphthyridine 7-oxide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1zzl | A | 6-[4-(4-fluorophenyl)-1,3-oxazol-5-yl]-3-isopropyl[1,2,4]triazolo[4,3-a]pyridine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3gfe | A | n-cyclopropyl-3-{[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-4-yl]amino}-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1bmk | A | 4-(fluorophenyl)-1-cyclopropylmethyl-5-(2-amino-4-pyrimidinyl)imidazole | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5n67 | A | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1r3c | A | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfk | A | B | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3iph | A | B | 6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3fly | A | 6-(2,4-difluorophenoxy)-8-methyl-2-[(1-methylethyl)amino]pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3lff | A | B | (4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acid | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfe | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-4-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6qdz | A | A | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh8 | A | A | [3-(benzyloxy)phenyl]methanol | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 8 | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfa | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2onl | B | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh1 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpt | A | B | n-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyy | A | 3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-4h-1,2,4-triazol-3-yl)phenol | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3d7z | A | A | n~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nww | A | 1-[2-(2-{[2-(dimethylamino)ethyl]amino}-6-{2-[(1-methylethyl)amino]-1,3-thiazol-5-yl}pyrimidin-4-yl)benzyl]-3-ethylurea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5wjj | A | B | n-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3huc | A | B | n-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3gc7 | A | B | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6zwp | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1oz1 | A | A | 3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-ol | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2baq | A | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvp | A | B | n-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3mgy | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfb | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnv | A | B | 1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylurea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zs5 | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv3 | A | A | 1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvm | A | 4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | A | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6zqs | A | 2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmm | A | 6-(2,4-difluorophenoxy)-n-[(1r)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fls | A | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3que | A | 2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfk | A | A | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3odz | X | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4fa2 | A | A | trans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanol | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3fc1 | X | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3e92 | A | n-cyclopropyl-2',6-dimethyl-4'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-3-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv4 | B | 1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbn | A | n-(3-tert-butyl-1h-pyrazol-5-yl)-n'-{4-chloro-3-[(pyridin-3-yloxy)methyl]phenyl}urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3roc | A | 3-{5-chloro-4-[(2,4-difluorobenzyl)oxy]-6-oxopyrimidin-1(6h)-yl}-n-(2-hydroxyethyl)-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcp | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv6 | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[4-(2-morpholin-4-ylethoxy)phenyl]urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2yiw | A | 1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwt | A | B | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnu | A | B | 2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | C | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh3 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcq | A | B | 1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 5 | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3l8x | A | n,4-dimethyl-3-[(1-phenyl-1h-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 8a8m | A | phosphomethylphosphonic acid adenosyl ester | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5etc | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1wfc | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4e6c | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1di9 | A | 4-[3-methylsulfanylanilino]-6,7-dimethoxyquinazoline | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3e93 | A | B | 4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | B | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsg | A | B | tak-715 | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | B | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6qyx | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3flz | A | 8-methyl-6-phenoxy-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3hub | A | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwv | A | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1yqj | A | 6((s)-3-benzylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyrazine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2npq | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 2 | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3new | A | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5o8u | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4e8a | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpa | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyx | A | B | n-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | A | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hvc | A | 4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4a9y | A | n-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh7 | A | A | (3-phenoxyphenyl)methanol | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3ody | X | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbo | A | 2-chlorophenol | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4r3c | A | B | 6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbw | A | 3-(1-naphthylmethoxy)pyridin-2-amine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvl | A | 4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 3 | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5a | X | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw5 | A | n-[2-(3-{[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]sulfanyl}-1h-indol-1-yl)ethyl]-3-(trifluoromethyl)benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3d83 | A | n-{4'-[(cyclopropylmethyl)carbamoyl]-6-methylbiphenyl-3-yl}-2-morpholin-4-ylpyridine-4-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6anl | A | A | tak-715 | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | C | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fsk | A | 3-(2-chlorophenyl)-7-[(trans-4-hydroxycyclohexyl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | C | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6zwp | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3lhj | A | n-cyclopropyl-3-[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-5-yl]-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4kip | B | 2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fl4 | A | 6-(2,4-difluorophenoxy)-3-(2-methylphenyl)-1h-pyrazolo[3,4-d]pyrimidine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3s4q | A | 3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-n-cyclopropyl-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3qud | A | B | {4-[(2-aminophenyl)amino]phenyl}(phenyl)methanone | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3gc7 | A | A | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh3 | A | naringenin | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvr | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwu | A | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1r39 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh2 | A | 3-phenylquinazolin-4(3h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2fsl | X | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2onl | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3ha8 | A | B | n~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvm | B | 4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3itz | A | 4-chloro-n-cyclopropyl-3-{[1-(2,6-difluorophenyl)-1h-pyrazolo[3,4-d]pyridazin-4-yl]amino}benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3kq7 | A | B | n-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6qe1 | A | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{r})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvp | A | A | n-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv4 | A | 1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3bx5 | A | n-[2-methyl-5-(methylcarbamoyl)phenyl]-2-{[(1r)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnw | A | A | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb1 | A | A | n-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9y | A | B | n,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3ocg | A | 5-amino-n-[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]-1-phenyl-1h-pyrazole-4-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2bal | A | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl][3-(piperidin-4-yloxy)phenyl]methanone | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5eta | B | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2fst | X | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv3 | A | B | 1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa0 | A | A | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2zaz | A | B | 4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehyde | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfc | A | (4-{5-[({4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}carbamoyl)amino]-3-tert-butyl-1h-pyrazol-1-yl}phenyl)acetic acid | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fln | C | 6-(2,4-difluorophenoxy)-8-methyl-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | B | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3gi3 | A | n-{5-tert-butyl-2-methoxy-3-[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]naphthalen-1-yl}carbamoyl)amino]phenyl}methanesulfonamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2fst | X | A | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | B | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1kv1 | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2i0h | A | B | 2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dione | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3pg3 | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa4 | A | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]furan-3-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbs | A | 3-fluoro-5-morpholin-4-yl-n-[3-(2-pyridin-4-ylethyl)-1h-indol-5-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1m7q | A | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperazin-1-yl-3,4-dihydroquinazolin-2(1h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | F | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4e6a | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3bv3 | A | 5-methyl-4-[(2-methyl-5-{[(3-morpholin-4-ylphenyl)carbonyl]amino}phenyl)amino]-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5mtx | A | A | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnx | A | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | B | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4l8m | A | A | n-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2bak | A | n-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfi | A | B | ~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2fsm | X | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsh | A | A | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | F | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hec | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3lff | A | A | (4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acid | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | B | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1w82 | A | n-[(3z)-5-tert-butyl-2-phenyl-1,2-dihydro-3h-pyrazol-3-ylidene]-n'-(4-chlorophenyl)urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4geo | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | D | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcs | A | A | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw7 | A | 2-({4-[(4-benzylpiperidin-1-yl)carbonyl]benzyl}sulfanyl)-3h-imidazo[4,5-c]pyridine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3d7z | A | B | n~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfo | A | A | 5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1ouk | A | 4-[5-[2-(1-phenyl-ethylamino)-pyrimidin-4-yl]-1-methyl-4-(3-trifluoromethylphenyl)-1h-imidazol-2-yl]-piperidine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3hl7 | A | 2-{4-[5-(4-chlorophenyl)-4-pyrimidin-4-yl-1h-pyrazol-3-yl]piperidin-1-yl}-2-oxoethanol | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6ohd | A | B | 3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4kip | A | 2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | C | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 9 | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hll | A | A | 3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4l8m | A | B | n-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3fml | A | 6-(2,4-difluorophenoxy)-n-[(1s)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmj | A | 4-(5-methyl-3-phenylisoxazol-4-yl)pyrimidin-2-amine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6m9l | A | 3-benzyl-6-[(2,4-difluorophenyl)amino]-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2y8o | A | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2zaz | A | A | 4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehyde | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1a9u | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3flq | A | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8t | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8p | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2yis | A | 1-[3-tert-butyl-1-(3-chloro-4-hydroxyphenyl)-1h-pyrazol-5-yl]-3-{2-[(3-{2-[(2-hydroxyethyl)sulfanyl]phenyl}[1,2,4]triazolo[4,3-a]pyridin-6-yl)sulfanyl]benzyl}urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp5 | A | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw6 | A | B | ethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylate | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2qd9 | A | 1-[(3ar)-5-{[3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8h)-yl]carbonyl}-6-methoxy-3ah-pyrrolo[2,3-b]pyridin-3-yl]-2-[(3r)-3-hydroxypyrrolidin-1-yl]-2-oxoethanone | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvl | B | 4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | A | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3iph | A | A | 6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwt | A | A | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3l8s | A | 3-[(4-bromo-2,6-difluorobenzyl)oxy]-5-{[(4-pyrrolidin-1-ylbutyl)carbamoyl]amino}isothiazole-4-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9w | A | B | n,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | H | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3fi4 | A | (2s)-1-{[3-(2-chlorophenyl)-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propan-2-ol | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8u | A | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3s3i | A | 3-(3-tert-butyl[1,2,4]triazolo[4,3-a]pyridin-7-yl)-n-cyclopropyl-4-methylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3dt1 | A | n-cyclopropyl-4-methyl-3-{2-[(2-morpholin-4-ylethyl)amino]quinazolin-6-yl}benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfd | A | 1-{4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcv | A | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1ouy | A | 1-(2,6-dichlorophenyl)-6-[(2,4-difluorophenyl)sulfanyl]-7-(1,2,3,6-tetrahydro-4-pyridinyl)-3,4-dihydropyrido[3,2-d]pyrimidin-2(1h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb1 | A | B | n-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5eta | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2yix | A | 1-ethyl-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3zs5 | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3rin | A | n-cyclopropyl-4-methyl-3-(2'-oxo-1',2'-dihydrospiro[cyclopentane-1,3'-indol]-6'-yl)benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbv | A | 3-fluoro-n-1h-indol-5-yl-5-morpholin-4-ylbenzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9y | A | A | n,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb0 | A | B | n-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnu | A | A | 2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zya | A | A | 2-amino-phenylamino-dibenzosuberone | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh7 | A | B | (3-phenoxyphenyl)methanol | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw6 | A | A | ethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylate | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2okr | D | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa5 | A | n-cyclopropyl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4fa2 | A | B | trans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanol | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwv | A | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3heg | A | B | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5n66 | A | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 1 | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | A | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6m95 | A | (4-benzylpiperidin-1-yl)[2-methoxy-4-(methylsulfanyl)phenyl]methanone | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 10 | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb0 | A | A | n-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6anl | A | B | tak-715 | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | D | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5ml5 | A | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-methylsulfanyl-1~{h}-imidazol-5-yl]pyridin-2-yl]propanamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 2rg6 | A | 4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methyl-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3ha8 | A | A | n~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 6 | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3e93 | A | A | 4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcs | A | B | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh6 | A | n-phenylpyridine-3-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3hll | A | B | 3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpt | A | A | n-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 7 | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyx | A | A | n-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | B | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 1kv2 | A | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmh | A | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3flw | A | 6-(2,4-difluorophenoxy)-2-{[3-hydroxy-1-(2-hydroxyethyl)propyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | D | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4ehv | A | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh0 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3hec | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1zz2 | A | n-[3-(4-fluorophenoxy)phenyl]-4-[(2-hydroxybenzyl)amino]piperidine-1-sulfonamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | B | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4ewq | A | B | 3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh4 | A | phenyl(piperidin-1-yl)methanone | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5etf | A | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3fkl | A | n-cyclopropyl-4-methyl-3-[8-methyl-7-oxo-2-(tetrahydro-2h-pyran-4-ylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh5 | A | benzyl pyridine-3-carboxylate | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5n67 | A | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4zth | A | A | 6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1zyj | A | 4-phenoxy-n-(pyridin-2-ylmethyl)benzamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3fkn | A | 3-[2-chloro-5-(methylsulfonyl)phenyl]-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | A | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | B | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 2rg5 | A | n-ethyl-4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5n65 | A | 2-phenyl-~{n}4-(2-thiophen-2-ylethyl)quinazoline-4,7-diamine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4dlj | A | 2-phenyl-n~4~-(2-phenylethyl)quinazoline-4,7-diamine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5n63 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcp | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1oz1 | A | B | 3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-ol | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsh | A | B | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6ohd | A | A | 3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcv | A | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5n64 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcq | A | A | 1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5omg | A | A | 3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | D | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa0 | A | B | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3pg3 | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | D | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3od6 | X | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5n68 | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsi | A | A | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5mz3 | A | A | ~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3new | A | B | - | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp2 | A | A | 1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-one | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 5eti | A | - | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 5omg | A | B | 3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmn | A | B | 6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvr | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}urea | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 1w7h | A | 3-(benzyloxy)pyridin-2-amine | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9w | A | A | n,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | Show | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw8 | A | 1-{4-[(1s)-1-amino-2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-(3-chloro-4-fluorophenyl)urea | Human | Show | | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | B | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | Show | |
