Aurora kinase A
Kinase structure
Kinase:AURKA (AurA)
Family:Aur
Group:Other
Species:HUMAN
IUPHAR/BPS ID:1936
PDB:6I2U
sc-PDB:
KIDFamMap:Search
Release date:2019-10-02
PubMed: 31546169
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):63.2° (19.1Å)
G-rich loop rotation:50.4°
Quality Score:8
Resolution:2.5 Å
Missing Residues:0
Missing Atoms:21
Ligand binding mode
Waters
Cluster
I7
I11
Ligand
No
No
Protein
Yes
No

Pocket alignment
Uniprot sequence:RPLGKGKFGNVYLLALKVLQLRREVEIQSHLRPNILRLYGYYLILEYAPLGTVYRELQKYCHSKRVIHRDIKPENLLLIADFGWS
Sequence structure:RPLGKGKFGNVYLLALKVLQLRREVEIQSHLRPNILRLYGYYLILEYAPLGTVYRELQKYCHSKRVIHRDIKPENLLLIADFGWS