Search results (276 entries covering 186 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
AURKA (AurA)AurOther8c1hAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther4uzdAethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHumanShow
AURKA (AurA)AurOther2wtvAA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther6c2tAB(2s,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-2-methyl-4-({3-[(1,3-thiazol-2-yl)amino]isoquinolin-1-yl}methyl)piperidine-4-carboxylic acidHumanShow
AURKA (AurA)AurOther3w2cE2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHumanShow
AURKA (AurA)AurOther3w10A1-(3-methoxyphenyl)-n-(5-methyl-1h-pyrazol-3-yl)isoquinolin-3-amineHumanShow
AURKA (AurA)AurOther4uynAethyl (9s)-9-[5-(1h-benzimidazol-2-ylsulfanyl)furan-2-yl]-8-hydroxy-5,6,7,9-tetrahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHumanShow
AURKA (AurA)AurOther2dwbAphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther5os5ABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3w2cC2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHumanShow
AURKA (AurA)AurOther6vpmABadenosine monophosphateHumanShow
AURKA (AurA)AurOther2c6eAn-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamideHumanShow
AURKA (AurA)AurOther5dn3ABadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther6vplBBphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther2wtvBA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther4dedA2-({2-[(4-carbamoylphenyl)amino]pyrimidin-4-yl}amino)benzamideHumanShow
AURKA (AurA)AurOther4j8nC-HumanShow
AURKA (AurA)AurOther3w2cG2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHumanShow
AURKA (AurA)AurOther3m11A1-(4-{2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHumanShow
AURKA (AurA)AurOther3mygA2-{ethyl[(5-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}isothiazol-3-yl)methyl]amino}-2-methylpropan-1-olHumanShow
AURKA (AurA)AurOther3e5aAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHumanShow
AURKA (AurA)AurOther3fdnAn-[3-(acetylamino)phenyl]-5-{(2e)-2-[(4-methoxyphenyl)methylidene]hydrazino}-3-methyl-1h-pyrazole-4-carboxamideHumanShow
AURKA (AurA)AurOther8c1iABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther8c1dABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther6z4yAB6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one HumanShow
AURKA (AurA)AurOther2xneA3-chloro-n-(4-morpholin-4-ylphenyl)-6-pyridin-3-ylimidazo[1,2-a]pyrazin-8-amineHumanShow
AURKA (AurA)AurOther6vpiABphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther5os5AAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5l8jABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther2bmcA(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther6c83Aphosphomethylphosphonic acid adenylate esterHumanShow
AURKA (AurA)AurOther3w16A4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2h)-oneHumanShow
AURKA (AurA)AurOther3uohA4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHumanShow
AURKA (AurA)AurOther4j8nB-HumanShow
AURKA (AurA)AurOther4j8nA-HumanShow
AURKA (AurA)AurOther5orvAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5dpvAB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther5dt0AB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther8of5Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther8jf4A2-[4-[4-[bis(oxidanylidene)-$l^5-sulfanyl]oxyphenyl]carbonylpiperazin-1-yl]-6-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-n-prop-2-ynyl-pyrimidine-4-carboxamideHumanShow
AURKA (AurA)AurOther5dnrAAadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther3efwB1-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHumanShow
AURKA (AurA)AurOther4deeAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5orrAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther4o0sAadenosineHumanShow
AURKA (AurA)AurOther6hjkA(~{e})-~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-but-2-enamideHumanShow
AURKA (AurA)AurOther7ayhA7-[2-[(4-methoxyphenyl)amino]pyrimidin-4-yl]-1,3,4,5-tetrahydro-1-benzazepin-2-oneHumanShow
AURKA (AurA)AurOther3h0zA4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHumanShow
AURKA (AurA)AurOther5odtAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther4ztqA(2z,5z)-2-[(4-ethylphenyl)imino]-3-(2-methoxyethyl)-5-(pyridin-4-ylmethylidene)-1,3-thiazolidin-4-oneHumanShow
AURKA (AurA)AurOther1ol6Aadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5odtABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5orwAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5g15AAphosphomethylphosphonic acid adenylate esterHumanShow
AURKA (AurA)AurOther2w1eA4-[(2-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-3-yl}-1h-benzimidazol-5-yl)methyl]morpholin-4-iumHumanShow
AURKA (AurA)AurOther2j50An-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHumanShow
AURKA (AurA)AurOther3h10D9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHumanShow
AURKA (AurA)AurOther5orzAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther7ficAA6-[(5-cyclopropyl-1~{h}-pyrazol-3-yl)amino]-2-[4-[(3-methyl-4-oxidanyl-phenyl)methyl]piperazin-1-yl]-~{n}-prop-2-ynyl-pyrimidine-4-carboxamideHumanShow
AURKA (AurA)AurOther8jmxA5-(4-morpholin-4-yl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2-oxidanyl-benzaldehydeHumanShow
AURKA (AurA)AurOther8sspABn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHumanShow
AURKA (AurA)AurOther8sspAAn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHumanShow
AURKA (AurA)AurOther4jbqAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHumanShow
AURKA (AurA)AurOther5dr2Aadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther3uo5A4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther2w1cA4-{[2-(4-{[(4-fluorophenyl)carbonyl]amino}-1h-pyrazol-3-yl)-1h-benzimidazol-6-yl]methyl}morpholin-4-iumHumanShow
AURKA (AurA)AurOther5os3Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5dr6AA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther3h0zC4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHumanShow
AURKA (AurA)AurOther7ztlABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther2j4zB4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHumanShow
AURKA (AurA)AurOther2j50Bn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHumanShow
AURKA (AurA)AurOther3vapA3-(1-{2-[(3-fluoropyridinium-4-yl)amino]-2-oxoethyl}-1h-pyrazol-4-yl)-6-methyl-8-[(3-{[(1r,3r)-3-methylpiperidinium-1-yl]methyl}-1,2-thiazol-5-yl)amino]imidazo[1,2-a]pyrazin-1-iumHumanShow
AURKA (AurA)AurOther6r4aAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther6vpmAAadenosine monophosphateHumanShow
AURKA (AurA)AurOther2wtvCA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther5osfAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5aagA[3-[[4-[6-chloranyl-2-(1,3-dimethylpyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl]pyrazol-1-yl]methyl]phenyl]-(4-methylpiperazin-1-yl)methanoneHumanShow
AURKA (AurA)AurOther5os1ABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5oneAB4-(propanoylamino)-~{n}-[4-[(5,8,11-trimethyl-6-oxidanylidene-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamideHumanShow
AURKA (AurA)AurOther7o2vA1-[[3,4-bis(fluoranyl)phenyl]methyl]-~{n}-[(1~{r})-2-[[(3~{e})-3-(1~{h}-imidazol-5-ylmethylidene)-2-oxidanylidene-1~{h}-indol-5-yl]amino]-2-oxidanylidene-1-phenyl-ethyl]-6-methyl-2-oxidanylidene-pyridine-3-carboxamideHumanShow
AURKA (AurA)AurOther4dhfB7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHumanShow
AURKA (AurA)AurOther5drdAadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther4bn1AAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther6vplABphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther5objAadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther3o50An-{3-methyl-4-[(3-pyrimidin-4-ylpyridin-2-yl)oxy]phenyl}-3-(trifluoromethyl)benzamideHumanShow
AURKA (AurA)AurOther5osdAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther6cpgD1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHumanShow
AURKA (AurA)AurOther6hjjAA~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-3-methyl-phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-butanamideHumanShow
AURKA (AurA)AurOther1muoAadenosineHumanShow
AURKA (AurA)AurOther5l8lABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3cohA8-ethyl-3,10,10-trimethyl-4,5,6,8,10,12-hexahydropyrazolo[4',3':6,7]cyclohepta[1,2-b]pyrrolo[2,3-f]indol-9(1h)-oneHumanShow
AURKA (AurA)AurOther8jg8A4-[5-[3-[bis(oxidanylidene)-$l^5-sulfanyl]oxyphenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-yl]morpholineHumanShow
AURKA (AurA)AurOther3uodA4-[(4-{[2-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzoic acidHumanShow
AURKA (AurA)AurOther2w1gA2-{4-[(cyclopropylcarbamoyl)amino]-1h-pyrazol-3-yl}-6-(morpholin-4-ium-4-ylmethyl)-1h-3,1-benzimidazol-3-iumHumanShow
AURKA (AurA)AurOther5orxAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther2x6eA6-bromo-7-{4-[(5-methylisoxazol-3-yl)methyl]piperazin-1-yl}-2-[4-(4-methylpiperazin-1-yl)phenyl]-1h-imidazo[4,5-b]pyridineHumanShow
AURKA (AurA)AurOther7ayiA7-(2-phenylazanylpyrimidin-4-yl)-1,3,4,5-tetrahydro-1-benzazepin-2-oneHumanShow
AURKA (AurA)AurOther2c6eBn-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamideHumanShow
AURKA (AurA)AurOther3uojB4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHumanShow
AURKA (AurA)AurOther4c3pDphosphomethylphosphonic acid adenylate esterHumanShow
AURKA (AurA)AurOther8ssoABn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHumanShow
AURKA (AurA)AurOther8ssoACn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHumanShow
AURKA (AurA)AurOther4j8nD-HumanShow
AURKA (AurA)AurOther3uo6B4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHumanShow
AURKA (AurA)AurOther4byiA(s)-n-((1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)methyl)acetamideHumanShow
AURKA (AurA)AurOther5aafA3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-n,n-dimethylbenzamideHumanShow
AURKA (AurA)AurOther5l8lAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3r21ABn-(2-aminoethyl)-n-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHumanShow
AURKA (AurA)AurOther5os4Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther2wtvBB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther5g1xAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5orpAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5g15ABphosphomethylphosphonic acid adenylate esterHumanShow
AURKA (AurA)AurOther5os2ABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3k5uA2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanolHumanShow
AURKA (AurA)AurOther5dpvAA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther6r4cAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3p9jA4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2h)-oneHumanShow
AURKA (AurA)AurOther5dt4Aadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther5dnrABadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther6c2tAA(2s,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-2-methyl-4-({3-[(1,3-thiazol-2-yl)amino]isoquinolin-1-yl}methyl)piperidine-4-carboxylic acidHumanShow
AURKA (AurA)AurOther4j8mA1-[4-[[4-[(5-cyclopentyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHumanShow
AURKA (AurA)AurOther5dt0AA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther6vpmBAadenosine monophosphateHumanShow
AURKA (AurA)AurOther8c1mAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther8c1fAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther8c1dAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther8c15ABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther8c14ABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3uojA4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHumanShow
AURKA (AurA)AurOther8pr7Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5orsAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther2c6dAAphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther2c6dABphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther1ol5Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther4zs0A5-hydroxy-1'h-1,2'-bibenzimidazol-2(3h)-oneHumanShow
AURKA (AurA)AurOther2wtwA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther4jboA1-(4-{2-[(6-{4-[2-(dimethylamino)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHumanShow
AURKA (AurA)AurOther1ol7Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3lauAn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]butanamideHumanShow
AURKA (AurA)AurOther5dr6AB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther4jbpA1-(4-{2-[(6-{4-[2-(4-hydroxypiperidin-1-yl)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHumanShow
AURKA (AurA)AurOther6vpjABphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther5aadA7-(1-benzyl-1h-pyrazol-4-yl)-6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridineHumanShow
AURKA (AurA)AurOther2bmcD(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther2x6dAA6-bromo-7-[4-(4-chlorobenzyl)piperazin-1-yl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3h-imidazo[4,5-b]pyridineHumanShow
AURKA (AurA)AurOther6vphABdithiane diolHumanShow
AURKA (AurA)AurOther6vpiAAphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther5lxmAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther6c2rAA(2r,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-4-({3-fluoro-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyridin-2-yl}methyl)-2-methylpiperidine-4-carboxylic acidHumanShow
AURKA (AurA)AurOther5ew9AB4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acidHumanShow
AURKA (AurA)AurOther3uolBn~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamineHumanShow
AURKA (AurA)AurOther2x6dAB6-bromo-7-[4-(4-chlorobenzyl)piperazin-1-yl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3h-imidazo[4,5-b]pyridineHumanShow
AURKA (AurA)AurOther7ztlAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5os6Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther6hjjAB~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-3-methyl-phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-butanamideHumanShow
AURKA (AurA)AurOther2xngABn-(3-{3-chloro-8-[(4-morpholin-4-ylphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzyl)methanesulfonamideHumanShow
AURKA (AurA)AurOther5dn3AAadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther2w1fAn-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamideHumanShow
AURKA (AurA)AurOther4byjA(s)-n-(1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)acetamideHumanShow
AURKA (AurA)AurOther5l8kAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3o51An-[4-({3-[5-fluoro-2-(methylideneamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-2-(phenylamino)benzamideHumanShow
AURKA (AurA)AurOther3uolAn~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamineHumanShow
AURKA (AurA)AurOther5os1AAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther6r4dAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3up7A2-({2-[(4-carboxyphenyl)amino]pyrimidin-4-yl}amino)benzoic acidHumanShow
AURKA (AurA)AurOther5aaeA3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-5-methylisoxazoleHumanShow
AURKA (AurA)AurOther5orzABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther4dhfA7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHumanShow
AURKA (AurA)AurOther5ortAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3h0zB4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHumanShow
AURKA (AurA)AurOther6vpgAAphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther2bmcE(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther4b0gAB6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridineHumanShow
AURKA (AurA)AurOther4prjAn-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHumanShow
AURKA (AurA)AurOther5oroAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3h10B9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHumanShow
AURKA (AurA)AurOther5ornAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther8ssoAAn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHumanShow
AURKA (AurA)AurOther5g1xABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther4jajAbenzo[c][1,8]naphthyridin-6(5h)-oneHumanShow
AURKA (AurA)AurOther5ew9AA4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acidHumanShow
AURKA (AurA)AurOther6vpjAAphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther5l8kABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3o50Bn-{3-methyl-4-[(3-pyrimidin-4-ylpyridin-2-yl)oxy]phenyl}-3-(trifluoromethyl)benzamideHumanShow
AURKA (AurA)AurOther5os0Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther2wtvDB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther4ztrA6-({4-[(z)-{(2z)-2-[(4-ethylphenyl)imino]-3-methyl-4-oxo-1,3-thiazolidin-5-ylidene}methyl]pyridin-2-yl}amino)pyridine-3-carboxylic acidHumanShow
AURKA (AurA)AurOther4uzdBethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHumanShow
AURKA (AurA)AurOther5orlAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3cohB8-ethyl-3,10,10-trimethyl-4,5,6,8,10,12-hexahydropyrazolo[4',3':6,7]cyclohepta[1,2-b]pyrrolo[2,3-f]indol-9(1h)-oneHumanShow
AURKA (AurA)AurOther6cpeAA-HumanShow
AURKA (AurA)AurOther3unzA4-({4-[(2-fluorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHumanShow
AURKA (AurA)AurOther8c1hABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther3uo4A4-{[4-(biphenyl-2-ylamino)pyrimidin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther6cpeAB-HumanShow
AURKA (AurA)AurOther3uohB4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHumanShow
AURKA (AurA)AurOther8c14AAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther2np8An-{3-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]phenyl}cyclopropanecarboxamideHumanShow
AURKA (AurA)AurOther3h10A9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHumanShow
AURKA (AurA)AurOther3uokB4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acidHumanShow
AURKA (AurA)AurOther6c2rAB(2r,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-4-({3-fluoro-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyridin-2-yl}methyl)-2-methylpiperidine-4-carboxylic acidHumanShow
AURKA (AurA)AurOther2xruA3-({[4-(4-methylpiperazin-1-yl)phenyl]carbonyl}amino)-n-[(1r)-1-phenylpropyl]-1h-thieno[3,2-c]pyrazole-5-carboxamideHumanShow
AURKA (AurA)AurOther3ha6An~2~-(3,4-dimethoxyphenyl)-n~4~-[2-(2-fluorophenyl)ethyl]-n~6~-quinolin-6-yl-1,3,5-triazine-2,4,6-triamineHumanShow
AURKA (AurA)AurOther6graA1-[(2~{r},3~{s})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{s})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{h}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)ureaHumanShow
AURKA (AurA)AurOther6r4bABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5dt3Aadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther7ficAB6-[(5-cyclopropyl-1~{h}-pyrazol-3-yl)amino]-2-[4-[(3-methyl-4-oxidanyl-phenyl)methyl]piperazin-1-yl]-~{n}-prop-2-ynyl-pyrimidine-4-carboxamideHumanShow
AURKA (AurA)AurOther6cpfAphosphomethylphosphonic acid adenylate esterHumanShow
AURKA (AurA)AurOther2wqeAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther8c1eAadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther8c1iAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther4b0gAA6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridineHumanShow
AURKA (AurA)AurOther4c3pAphosphomethylphosphonic acid adenylate esterHumanShow
AURKA (AurA)AurOther6vplAAphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther8c1kAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5l8jAAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther4deaA4,4'-(pyrimidine-2,4-diyldiimino)dibenzoic acidHumanShow
AURKA (AurA)AurOther3nrmAn-(3-methylisothiazol-5-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-amineHumanShow
AURKA (AurA)AurOther3unzB4-({4-[(2-fluorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHumanShow
AURKA (AurA)AurOther3qbnA5-chloro-n~4~-cyclopropyl-n~2~-[4-(2-methoxyethoxy)phenyl]pyrimidine-2,4-diamineHumanShow
AURKA (AurA)AurOther2bmcB(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther2wtvCB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther5dosAadenosine-5'-triphosphateHumanShow
AURKA (AurA)AurOther3uo6A4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHumanShow
AURKA (AurA)AurOther6z4yAA6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one HumanShow
AURKA (AurA)AurOther5oneAA4-(propanoylamino)-~{n}-[4-[(5,8,11-trimethyl-6-oxidanylidene-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamideHumanShow
AURKA (AurA)AurOther2bmcF(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther3up2A4-[(4-{[2-(trifluoromethoxy)phenyl]amino}pyrimidin-2-yl)amino]benzoic acidHumanShow
AURKA (AurA)AurOther3efwA1-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHumanShow
AURKA (AurA)AurOther6cpgA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHumanShow
AURKA (AurA)AurOther2x81A4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther8guwAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther2bmcC(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHumanShow
AURKA (AurA)AurOther6vplBAphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther5dr9A4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther4bn1ABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5zanA7-(4-methylpiperazin-1-yl)-n-(5-methyl-1h-pyrazol-3-yl)-2-[(e)-2-phenylethenyl]quinazolin-4-amineHumanShow
AURKA (AurA)AurOther5oseAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther2xngAAn-(3-{3-chloro-8-[(4-morpholin-4-ylphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzyl)methanesulfonamideHumanShow
AURKA (AurA)AurOther3w2cA2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHumanShow
AURKA (AurA)AurOther8c1gAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5oryAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther2wtvAB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther3w18B2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamideHumanShow
AURKA (AurA)AurOther4debA4-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzamideHumanShow
AURKA (AurA)AurOther3r22An-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHumanShow
AURKA (AurA)AurOther5lxmABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther6xkaA-HumanShow
AURKA (AurA)AurOther2j4zA4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHumanShow
AURKA (AurA)AurOther6vphAAdithiane diolHumanShow
AURKA (AurA)AurOther3w18A2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamideHumanShow
AURKA (AurA)AurOther6r49Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther6vpmBBadenosine monophosphateHumanShow
AURKA (AurA)AurOther8c1fABadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther4cegAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther5obrA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHumanShow
AURKA (AurA)AurOther4o0wAadenosineHumanShow
AURKA (AurA)AurOther3r21AAn-(2-aminoethyl)-n-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHumanShow
AURKA (AurA)AurOther4ztsA(2z,5z)-2-[(4-ethylphenyl)imino]-3-methyl-5-[(2-{[4-(1h-tetrazol-5-yl)phenyl]amino}pyridin-4-yl)methylidene]-1,3-thiazolidin-4-oneHumanShow
AURKA (AurA)AurOther6i2uA-HumanShow
AURKA (AurA)AurOther3h0yA2-chloro-n-[4-({5-fluoro-2-[(4-hydroxyphenyl)amino]pyrimidin-4-yl}amino)phenyl]benzamideHumanShow
AURKA (AurA)AurOther4uzhA(4s)-4-(2-fluorophenyl)-2,4,6,7,8,9-hexahydro-5h-pyrazolo[3,4-b][1,7]naphthyridin-5-oneHumanShow
AURKA (AurA)AurOther6c83Bphosphomethylphosphonic acid adenylate esterHumanShow
AURKA (AurA)AurOther6vpgABphosphoaminophosphonic acid-adenylate esterHumanShow
AURKA (AurA)AurOther4o0uAadenosineHumanShow
AURKA (AurA)AurOther3uokA4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acidHumanShow
AURKA (AurA)AurOther2w1dA2-(1h-pyrazol-3-yl)-1h-benzimidazoleHumanShow
AURKA (AurA)AurOther2wtvDA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHumanShow
AURKA (AurA)AurOther8c15AAadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther4c3rAphosphomethylphosphonic acid adenylate esterHumanShow
AURKA (AurA)AurOther1mq4Aadenosine-5'-diphosphateHumanShow
AURKA (AurA)AurOther4jaiAn-{4-[(6-oxo-5,6-dihydrobenzo[c][1,8]naphthyridin-1-yl)amino]phenyl}benzamideHumanShow
AURKA (AurA)AurOther5os2AAadenosine-5'-diphosphateHumanShow