P21 protein (Cdc42/Rac)-activated kinase 4
Kinase structure
Kinase:PAK4
Family:STE20
Group:STE
Species:HUMAN
IUPHAR/BPS ID:2136
PDB:6WLY
sc-PDB:
KIDFamMap:Search
Release date:2020-06-24
PubMed: 32585314
Chain:A
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 6WLY
6WLYAlternative model: AChain: A
6WLYAlternative model: CChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):50.1° (15Å)
G-rich loop rotation:64°
Quality Score:9.5
Resolution:1.9 Å
Missing Residues:0
Missing Atoms:5
Ligand binding mode
Waters
Cluster
I1
I2
I3
I4
Ligand
No
No
No
No
Protein
Yes
No
Yes
Yes

Pocket alignment
Uniprot sequence:IKIGEGSTGIVCIVAVKKMLLFNEVVIMRDYQENVVEMYNSWVVMEFLEGGALTDIVTHVLHAQGVIHRDIKSDSILLLSDFGFC
Sequence structure:IKIGEGSTGIVCIVAVKKMLLFNEVVIMRDYQENVVEMYNSWVVMEFLEGGALTDIVTHVLHAQGVIHRDIKSDSILLLSDFGFC