MER proto-oncogene, tyrosine kinase
Kinase structure
Kinase:MERTK (MER)
Family:Axl
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1837
PDB:7AB0
sc-PDB:
KIDFamMap:Search
Release date:2020-10-28
PubMed: 33119085
Chain:A
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 7AB0
7AB0Alternative model: AChain: A


Structural information
DFG conformation:in
αC-helix conformation:out
G-rich loop angle (distance):58.8° (18.6Å)
G-rich loop rotation:29.1°
Quality Score:7.8
Resolution:1.74 Å
Missing Residues:3
Missing Atoms:10
Ligand binding mode
Waters
Cluster
I1
I4
I5
I8
Ligand
No
No
No
No
Protein
Yes
No
Yes
No

Pocket alignment
Uniprot sequence:KILGEGEFGSVMEVAVKTMEFLSEAACMKDFSPNVIRLLGVMVILPFMKYGDLHTYLLYYLSNRNFLHRDLAARNCMLVADFGLS
Sequence structure:RILGEGEFGSVMEVAVKTMEFLSEAACMKDFSPNVIRLLGVMVILPFMKYGDLHTYLLYYLSNRNFLHRDLAARNCMLVADF___