Checkpoint kinase 1
Kinase structure
Kinase:CHEK1 (CHK1)
Family:CAMKL
Group:CAMK
Species:HUMAN
IUPHAR/BPS ID:1987
PDB:7AKM
sc-PDB:
KIDFamMap:Search
Release date:2021-04-14
PubMed: 33789090
Chain:B
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 7AKM
7AKMAlternative model: AChain: A
7AKMAlternative model: AChain: B
7AKMAlternative model: BChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):60.5° (18Å)
G-rich loop rotation:52.9°
Quality Score:8
Resolution:1.93 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I3
I4
I5
I6
I9
I11
Ligand
No
No
No
No
No
No
Protein
Yes
Yes
Yes
No
No
Yes

Pocket alignment
Uniprot sequence:QTLGEGAYGEVQLVAVKIVNIKKEICINKMLNENVVKFYGHYLFLEYCSGGELFDRIEPYLHGIGITHRDIKPENLLLISDFGLA
Sequence structure:QTLGEGAYGEVQLVAVKIVNIKKEICINKMLNENVVKFYGHYLFLEYCSGGELFDRIEPYLHGIGITHRDIKPENLLLISDFGLA