PDB-code
Search results (237 entries covering 158 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
 | CHEK1 (CHK1) | CAMKL | CAMK | 4ft5 | A | B | 1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | Show |  |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmt | A | A | 2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ywp | A | 1-(5-chloro-2,4-dimethoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsw | A | B | 8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym6 | A | A | 1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fcf | A | A | 4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hxl | A | 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)-1h-indazole-6-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgx | A | 2-[(6-amino-7h-purin-8-yl)thio]acetamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3f9n | A | B | - | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yer | A | B | 5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op4 | A | [4-[[4-(ethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-fluoranyl-5-methoxy-phenyl]-morpholin-4-yl-methanone | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmv | A | 1-[(2s)-4-(7h-purin-6-yl)morpholin-2-yl]methanamine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftk | A | A | 3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftr | A | B | 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyi | A | B | 2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fti | A | B | methyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | A | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsw | A | A | 8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmw | A | 1-[(2s)-4-(5-bromo-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydk | A | 2-(carbamoylamino)-5-phenyl-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1zlt | A | (4z)-4-(2-amino-5-oxo-3,5-dihydro-4h-imidazol-4-ylidene)-2,3-dichloro-4,5,6,7-tetrahydropyrrolo[2,3-c]azepin-8(1h)-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq6 | A | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brn | A | (2r)-1-[(5,6-diphenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]propan-2-ol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opb | A | A | (2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftn | A | A | 4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opv | A | 4-(3-methylphenyl)-6-[(1-methylpyrazol-3-yl)amino]-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsu | A | B | 4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydj | B | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjj | A | B | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym4 | A | B | ethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmq | A | n-(4-oxo-5,6,7,8-tetrahydro-4h-[1,3]thiazolo[5,4-c]azepin-2-yl)acetamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | A | B | staurosporine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op2 | A | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyf | A | 4-[3-amino-6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acid | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4gh2 | A | B | 3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hog | A | (5-{3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-1h-indazol-6-yl}-2h-1,2,3-triazol-4-yl)methanol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsq | A | B | 4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brg | A | (5,6-diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-acetic | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjd | A | B | 2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym6 | A | B | 1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft3 | A | A | 1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylurea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qye | A | 4-[6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acid | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa4 | A | B | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftl | A | B | 4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9n | A | 3-(4'-hydroxybiphenyl-4-yl)-n-(4-hydroxycyclohexyl)-1,4-dihydroindeno[1,2-c]pyrazole-6-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk1 | A | 4-amino-2-[(1,3-dimethyl-1h-pyrazol-4-yl)amino]-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftq | A | A | 5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym3 | A | B | ethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot3 | A | B | 5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot3 | A | A | 5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opu | A | 6-azanyl-4-(3-methylphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym3 | A | A | ethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5dls | A | 1-benzyl-n-(5-{5-[3-(dimethylamino)-2,2-dimethylpropoxy]-1h-indol-2-yl}-6-oxo-1,6-dihydropyridin-3-yl)-1h-pyrazole-4-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1zys | A | n-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}nicotinamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftt | A | B | methyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmt | A | B | 2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa4 | A | A | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydi | A | A | 5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fck | A | A | 2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvs | A | rel-(9r,12s)-9,10,11,12-tetrahydro-9,12-epoxy-1h-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-1,3(2h)-dione | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvm | A | 3-[4-(piperidin-1-ylmethyl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8siw | A | (1s,2s)-n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)-2-(1-methyl-1h-pyrazol-4-yl)cyclopropane-1-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft0 | A | A | 2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9v | B | 18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ghg | A | 5-{5-[(s)-2-amino-3-(1h-indol-3-yl)-propoxyl]-pyridin-3-yl}-3-[1-(1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opb | A | B | (2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9p | A | 1-(5-chloro-2-methoxyphenyl)-3-{6-[2-(dimethylamino)-1-methylethoxy]pyrazin-2-yl}urea | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyh | A | B | 2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftt | A | A | methyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftq | A | B | 5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk3 | A | 4-amino-7-methyl-2-({5-methyl-1-[(3s)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot8 | A | B | n-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgv | A | (2s)-1-amino-3-[(5-nitroquinolin-8-yl)amino]propan-2-ol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5f4n | A | B | methyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fto | A | B | 4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fst | A | A | 4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bko | A | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftk | A | B | 3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op7 | A | [4-[[5-chloranyl-4-(methylamino)-7~{h}-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxy-phenyl]-morpholin-4-yl-methanone | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsz | A | A | (3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3k | A | 4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-2-methoxyphenol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | B | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftc | A | B | 1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)urea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | A | A | phosphothiophosphoric acid-adenylate ester | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9v | A | 18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hxq | A | 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)quinolin-2(1h)-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvr | A | staurosporine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmu | A | A | 6-morpholin-4-yl-9h-purine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftn | A | B | 4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsu | A | A | 4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2bro | A | (2r)-3-{[(4z)-5,6-diphenyl-6,7-dihydro-4h-pyrrolo[2,3-d]pyrimidin-4-ylidene]amino}propane-1,2-diol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydj | A | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym4 | A | A | ethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym8 | A | (r)-5-(8-chloroisoquinolin-3-ylamino)-3-(1-(dimethylamino)propan-2-yloxy)pyrazine-2-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk2 | A | 4-amino-7-methyl-2-({5-methyl-1-[(3r)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3nlb | A | 3-methyl-5-[5-(1-methylethyl)-1h-benzimidazol-2-yl]-n-(1-methylpiperidin-4-yl)-1h-pyrazole-4-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4jik | A | 2-(4-chlorophenyl)-8-[(3s)-piperidin-3-ylamino]imidazo[1,2-c]pyrimidine-5-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyh | B | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym5 | A | (3-{4-[(2s)-2-(aminomethyl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}phenyl)methanol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8e80 | A | 2-[(1r,4r)-2-{(6p)-6-[(6m)-6-(1h-pyrazol-5-yl)-1h-indazol-1-yl]pyrimidin-4-yl}-2-azabicyclo[2.1.1]hexan-4-yl]propan-2-ol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmx | A | 1-[(2s)-4-(5-phenyl-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | A | A | staurosporine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brb | A | 2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fta | A | B | 6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjx | A | B | 4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyg | A | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acid | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | A | B | phosphothiophosphoric acid-adenylate ester | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft9 | A | A | 1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylurea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | B | A | staurosporine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | B | B | - | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yex | A | A | 5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft9 | A | B | 1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylurea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4gh2 | A | A | 3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | A | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3l | A | 3-(1h-benzimidazol-2-yl)-1h-indazole | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyg | B | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acid | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op2 | A | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsy | A | A | 2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fc8 | A | A | 2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bkn | A | adenine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3tki | A | n-(2-aminoethyl)-5-(2-{[4-(morpholin-4-yl)pyridin-2-yl]amino}-1,3-thiazol-5-yl)pyridine-3-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgu | A | 2,2'-{[9-(hydroxyimino)-9h-fluorene-2,7-diyl]bis(oxy)}diacetic acid | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq5 | A | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | B | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjm | A | 4-amino-6-{[(2-fluorophenyl)methyl]amino}-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | B | A | - | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjh | A | B | n,n-dimethyl-7h-purin-6-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8siv | A | n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)cyclopropanecarboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3j | A | debromohymenialdisine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjx | A | A | 4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8e81 | A | (1s)-1-[(1p)-1-{6-[(3r)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}-1h-indazol-6-yl]spiro[2.2]pentane-1-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot8 | A | A | n-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fcf | A | B | 4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yex | A | B | 5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvk | A | n-[3-(6-cyano-9h-pyrrolo[2,3-b:5,4-c']dipyridin-3-yl)phenyl]acetamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sug | A | A | 1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2br1 | A | A | 2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bje | A | B | adenine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa3 | A | A | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brm | A | B | 3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft5 | A | A | 1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydi | A | B | 5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsq | A | A | 4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym7 | A | B | 5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8i | A | A | 7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5f4n | A | A | methyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op5 | A | 3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym7 | A | A | 5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftl | A | A | 4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-ol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsr | A | A | 6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazole | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | C | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brm | A | A | 3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | A | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9o | A | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5ops | A | 4-(3-hydroxyphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjd | A | A | 2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsn | A | A | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2r0u | A | 6-(3-aminopropyl)-4-(3-hydroxyphenyl)-9-(1h-pyrazol-4-yl)benzo[h]isoquinolin-1(2h)-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xf0 | A | 3-phenyl-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjh | A | A | n,n-dimethyl-7h-purin-6-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fti | A | A | methyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suf | A | A | 8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oor | A | staurosporine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftr | A | A | 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft7 | A | B | 1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8six | A | (1s)-n-(7-chloro-6-{4-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperazin-1-yl}isoquinolin-3-yl)-6-oxaspiro[2.5]octane-1-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fck | A | B | 2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2qhn | A | 5-ethyl-3-methyl-1,5-dihydro-4h-pyrazolo[4,3-c]quinolin-4-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq8 | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftj | A | A | trans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyh | A | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fc8 | A | B | 2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xez | A | 6-(1h-pyrazol-3-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | B | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa5 | A | B | 2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjj | A | A | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suj | A | (3r,4r)-4-{4-[6-chloro-2-({1-[(1r)-2,2-difluorocyclopropyl]-5-methyl-1h-pyrazol-4-yl}amino)quinazolin-7-yl]piperidin-1-yl}-4-methyloxolan-3-ol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3jvs | A | - | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft3 | A | B | 1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylurea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brh | A | A | n-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sug | A | B | 1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suh | A | 1-[5-chloro-4-({6-chloro-7-[1-(oxetan-3-yl)piperidin-4-yl]quinazolin-2-yl}amino)-1h-pyrazol-1-yl]-2-methylpropan-2-ol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3jvr | A | - | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa3 | A | B | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fst | A | B | 4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ayp | A | (3z)-6-(4-hydroxy-3-methoxyphenyl)-3-(1h-pyrrol-2-ylmethylene)-1,3-dihydro-2h-indol-2-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmu | A | B | 6-morpholin-4-yl-9h-purine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8d | A | B | 5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fto | A | A | 4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrile | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oot | A | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1ia8 | A | - | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsm | A | B | 4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3f9n | A | A | - | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsn | A | B | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsm | A | A | 4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2qhm | A | (3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl 1h-pyrrolo[2,3-b]pyridine-3-carboxylate | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjr | A | 4-amino-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3tkh | A | 1-(morpholin-4-yl)-2-[4-(2-{[5-(pyridin-3-yl)-1,3-thiazol-2-yl]amino}pyridin-4-yl)piperazin-1-yl]ethanone | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvl | A | 3-(2-hydroxyphenyl)-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftu | A | B | methyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsz | A | B | (3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7mck | A | n-{5-[(3s)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(trifluoromethyl)pyridin-3-yl}-6-(1-methyl-1h-pyrazol-4-yl)pyridine-2-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oop | A | A | phosphoaminophosphonic acid-adenylate ester | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsy | A | B | 2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fta | A | A | 6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wms | A | [4-amino-2-(tert-butylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsr | A | B | 6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazole | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftj | A | B | trans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftc | A | A | 1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)urea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9u | A | 18-chloro-11,12,13,14-tetrahydro-1h,10h-8,4-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecin-2-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yer | A | A | 5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftu | A | A | methyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyh | A | A | 2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft7 | A | A | 1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brh | A | B | n-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgw | A | 4,4'-(1-propyl-1h-1,2,4-triazole-3,5-diyl)bis(2,5-dihydro-1,2,5-oxadiazol-3-amine) | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2br1 | A | B | 2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8i | A | B | 7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmr | A | B | 5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa5 | A | A | 2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjo | A | 4-amino-6-(2,3-difluorophenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oop | A | B | phosphoaminophosphonic acid-adenylate ester | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xey | A | 3-(1h-indol-3-yl)-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3u9n | A | 2-(2,3-dihydro-1-benzofuran-5-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | B | B | staurosporine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sui | A | (3r,4r)-4-{(3s,4s)-4-[6-chloro-2-({5-chloro-1-[(1r)-2,2-difluorocyclopropyl]-1h-pyrazol-4-yl}amino)quinazolin-7-yl]-3-fluoropiperidin-1-yl}oxolan-3-ol | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvq | A | 7-hydroxystaurosporine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opr | A | 5-[4-(morpholin-4-ylmethyl)phenyl]-3-(1-propan-2-yl-1,2,3-triazol-4-yl)pyridin-2-amine | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft0 | A | B | 2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acid | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmr | A | A | 5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-one | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2gdo | A | 4-[(3s)-1-azabicyclo[2.2.2]oct-3-ylamino]-3-(1h-benzimidazol-2-yl)-6-chloroquinolin-2(1h)-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bje | A | A | adenine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyi | A | A | 2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hy0 | A | 3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-6-(1h-pyrazol-4-yl)quinolin-2(1h)-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8e | A | 5-methyl-8-pyridin-4-yl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suf | A | B | 8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amine | Human | Show | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8d | A | A | 5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | Show | |
