P21 protein (Cdc42/Rac)-activated kinase 4
Kinase structure
Kinase:PAK4
Family:STE20
Group:STE
Species:HUMAN
IUPHAR/BPS ID:2136
PDB:2Q0N
sc-PDB:
KIDFamMap:Search
Release date:2007-06-26
Chain:A
(Alternate) Model:A
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The orthosteric binding pocket


More entries for 2Q0N
2Q0NAlternative model: BChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):52.1° (15.7Å)
G-rich loop rotation:56.8°
Quality Score:9.7
Resolution:1.75 Å
Missing Residues:0
Missing Atoms:3
Ligand binding mode
Waters
Cluster
I1
I2
I3
I5
I6
I9
Ligand
No
No
No
No
No
No
Protein
Yes
No
Yes
Yes
No
No

Pocket alignment
Uniprot sequence:IKIGEGSTGIVCIVAVKKMLLFNEVVIMRDYQENVVEMYNSWVVMEFLEGGALTDIVTHVLHAQGVIHRDIKSDSILLLSDFGFC
Sequence structure:IKIGEGSTGIVCIVAVKKMLLFNEVVIMRDYQENVVEMYNSWVVMEFLEGGALTDIVTHVLHAQGVIHRDIKSDSILLLSDFGFC