Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Kinase structure
Kinase:PIK3CA (p110a)
Family:PIK
Group:Atypical
Species:HUMAN
IUPHAR/BPS ID:2153
PDB:7MYN
sc-PDB:
KIDFamMap:Search
Release date:2021-11-10
PubMed: 34725156
Chain:A
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 7MYN
7MYNAlternative model: AChain: A


Structural information
DFG conformation:out-like
αC-helix conformation:in
G-rich loop angle (distance):56.2° (17Å)
G-rich loop rotation:83.9°
Quality Score:8
Resolution:2.79 Å
Missing Residues:0
Missing Atoms:0

Pocket alignment
Uniprot sequence:CRIMSSAKRPLWLIIFKNGDLRQDMLTLQIIRLRMLPYGCLVGLIEVVRSHTIMQIQCKATFI--LGIGDRHNSNIMVHIDFGHF
Sequence structure:CRIMSSAKRPLWLIIFKNGDLRQDMLTLQIIRLRMLPYGCLVGLIEVVRSHTIMQIQCKATFI__LGIGDRHNSNIMVHIDFGHF