P21 protein (Cdc42/Rac)-activated kinase 4
Kinase structure
Kinase:PAK4
Family:STE20
Group:STE
Species:HUMAN
IUPHAR/BPS ID:2136
PDB:4FIH
sc-PDB:
KIDFamMap:Search
Release date:2012-09-12
PubMed: 22988085
Chain:A
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 4FIH
4FIHAlternative model: AChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):49.5° (14.8Å)
G-rich loop rotation:65.8°
Quality Score:8
Resolution:1.97 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I2
I3
I4
I7
I8
I9
Ligand
No
No
No
No
No
No
No
Protein
Yes
No
No
Yes
No
Yes
No

Pocket alignment
Uniprot sequence:IKIGEGSTGIVCIVAVKKMLLFNEVVIMRDYQENVVEMYNSWVVMEFLEGGALTDIVTHVLHAQGVIHRDIKSDSILLLSDFGFC
Sequence structure:IKIGEGSTGIVCIVAVKKMLLFNEVVIMRDYQENVVEMYNSWVVMEFLEGGALTDIVTHVLHAQGVIHRDIKSDSILLLSDFGFC