P21 protein (Cdc42/Rac)-activated kinase 1
Kinase structure
Kinase:PAK1
Family:STE20
Group:STE
Species:HUMAN
IUPHAR/BPS ID:2133
PDB:4O0R
sc-PDB:
KIDFamMap:Search
Release date:2014-02-12
PubMed: 24432870
Chain:B
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The orthosteric binding pocket


More entries for 4O0R
4O0RChain: A


Structural information
DFG conformation:in
αC-helix conformation:out
G-rich loop angle (distance):69.4° (19.9Å)
G-rich loop rotation:52.1°
Quality Score:7.2
Resolution:2.4 Å
Missing Residues:2
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I7
Ligand
No
Protein
Yes

Pocket alignment
Uniprot sequence:EKIGQGASGTVYTVAIKQMLIINEILVMRENKPNIVNYLDSWVVMEYLAGGSLTDVVTEFLHSNQVIHRDIKSDNILLLTDFGFC
Sequence structure:EKIGQGASGTVYTVAIKQMLIINEILVMRENKPNIVNYLDSWVVMEYLAGGSLTDVVTEFLHSNQVIHRNIKSDNILLLTDFG__