KIT proto-oncogene receptor tyrosine kinase
Kinase structure
Kinase:KIT
Family:PDGFR
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1805
PDB:8DFM
sc-PDB:
KIDFamMap:Search
Release date:2023-03-29
PubMed: 36943885
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:out-like
αC-helix conformation:out
G-rich loop angle (distance):108.9° (49.8Å)
G-rich loop rotation:104.7°
Quality Score:2
Resolution:3.45 Å
Missing Residues:5
Missing Atoms:53

Pocket alignment
Uniprot sequence:KTLGAGAFGKVVEVAVKMLALMSELKVLSYLGMNIVNLLGALVITEYCCYGDLLNFLRRFLASKNCIHRDLAARNILLICDFGLA
Sequence structure:AEANTGK_YTVFVKLFDLVREVYSKFIGICL_SD__QEGSFILYSKQEKSWHHDISSANVMCVGI_