P21 protein (Cdc42/Rac)-activated kinase 1
Kinase structure
Kinase:PAK1
Family:STE20
Group:STE
Species:HUMAN
IUPHAR/BPS ID:2133
PDB:8X5Z
sc-PDB:
KIDFamMap:Search
Release date:2023-12-06
Chain:A
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 8X5Z
8X5ZAlternative model: AChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):-
G-rich loop rotation:-
Quality Score:6.8
Resolution:1.8 Å
Missing Residues:3
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I2
I4
I6
I8
Ligand
No
No
No
No
No
Protein
No
No
Yes
No
Yes

Pocket alignment
Uniprot sequence:EKIGQGASGTVYTVAIKQMLIINEILVMRENKPNIVNYLDSWVVMEYLAGGSLTDVVTEFLHSNQVIHRDIKSDNILLLTDFGFC
Sequence structure:EKIGQ___GTVYTVAIRQMLIINEILVMRENKPNIVNYLDSWVVMEYLAGGSLTDVVTEFLHSNQVIHRDIKSDNILLLTDFGFC