Fibroblast growth factor receptor 4
Kinase structure
Kinase:FGFR4
Family:FGFR
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1811
PDB:8KH9
sc-PDB:
KIDFamMap:Search
Release date:2024-07-31
PubMed: 38348819
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):57.4° (16.6Å)
G-rich loop rotation:55.1°
Quality Score:9.2
Resolution:1.42 Å
Missing Residues:0
Missing Atoms:8
Ligand binding mode
Waters
Cluster
I4
I5
I10
Ligand
No
No
No
Protein
Yes
Yes
Yes

Pocket alignment
Uniprot sequence:KPLGEGCFGQVVRVAVKMLDLVSEMEVMKLIGKNIINLLGVYVIVECAAKGNLREFLRAYLESRKCIHRDLAARNVLVIADFGLA
Sequence structure:KPLGEGAFGQVVRVAVKMLDLVSEMEVMKLIGKNIINLLGVYVIMECAAKGNLREFLRAYLESRKCIHRDLAARNVLVIADFGLA