P21 protein (Cdc42/Rac)-activated kinase 1
Kinase structure
Kinase:PAK1
Family:STE20
Group:STE
Species:HUMAN
IUPHAR/BPS ID:2133
PDB:1F3M
sc-PDB:
KIDFamMap:Search
Release date:2000-06-29
PubMed: 10975528
Chain:D
Click to open a 3D viewer
The orthosteric binding pocket


More entries for 1F3M
1F3MChain: C


Structural information
DFG conformation:in
αC-helix conformation:out
G-rich loop angle (distance):80.6° (23.5Å)
G-rich loop rotation:37.6°
Quality Score:7.6
Resolution:2.3 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I6
Ligand
No
Protein
No

Pocket alignment
Uniprot sequence:EKIGQGASGTVYTVAIKQMLIINEILVMRENKPNIVNYLDSWVVMEYLAGGSLTDVVTEFLHSNQVIHRDIKSDNILLLTDFGFC
Sequence structure:EKIGQGASGTVYTVAIRQMLIINEILVMRENKPNIVNYLDSWVVMEYLAGGSLTDVVTEFLHSNQVIHRDIKSDNILLLTDFGFC