Adrenergic, beta, receptor kinase 1
Kinase structure
Kinase:GRK2 (BARK1)
Family:GRK
Group:AGC
Species:HUMAN
IUPHAR/BPS ID:1466
PDB:3CIK
sc-PDB:
KIDFamMap:Search
Release date:2009-02-17
PubMed: 20128603
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):62.7° (18.4Å)
G-rich loop rotation:69.5°
Quality Score:8
Resolution:2.75 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I5
Ligand
No
Protein
Yes

Pocket alignment
Uniprot sequence:RIIGRGGFGEVYGYAMKCLLALNERIMLSLVSPFIVCMSYASFILDLMNGGDLHYHLSQHMHNRFVVYRDLKPANILLISDLGLA
Sequence structure:RIIGRGGFGEVYGYAMKCLLALNERIMLSLVSPFIVCMSYASFILDLMNGGDLHYHLSQHMHNRFVVYRDLKPANILLISDLGLA