P21 protein (Cdc42/Rac)-activated kinase 1
Kinase structure
Kinase:PAK1
Family:STE20
Group:STE
Species:HUMAN
IUPHAR/BPS ID:2133
PDB:1YHV
sc-PDB:
KIDFamMap:Search
Release date:2005-05-24
PubMed: 15893667
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):66.5° (20Å)
G-rich loop rotation:37.8°
Quality Score:9.5
Resolution:1.8 Å
Missing Residues:0
Missing Atoms:5
Ligand binding mode
Waters
Cluster
I1
I2
I4
I5
I6
I8
Ligand
No
No
No
No
No
No
Protein
Yes
Yes
Yes
No
Yes
Yes

Pocket alignment
Uniprot sequence:EKIGQGASGTVYTVAIKQMLIINEILVMRENKPNIVNYLDSWVVMEYLAGGSLTDVVTEFLHSNQVIHRDIKSDNILLLTDFGFC
Sequence structure:EKIGQGASGTVYTVAIRQMLIINEILVMRENKPNIVNYLDSWVVMEYLAGGSLTDVVTEFLHSNQVIHRDIKSDNILLLTDFGFC