P21 protein (Cdc42/Rac)-activated kinase 1
Kinase structure
Kinase:PAK1
Family:STE20
Group:STE
Species:HUMAN
IUPHAR/BPS ID:2133
PDB:3Q4Z
sc-PDB:
KIDFamMap:Search
Release date:2011-12-21
PubMed: 22153498
Chain:B
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 3Q4Z
3Q4ZAlternative model: AChain: A
3Q4ZAlternative model: AChain: B
3Q4ZAlternative model: BChain: A


Structural information
DFG conformation:in
αC-helix conformation:out
G-rich loop angle (distance):70.5° (19.9Å)
G-rich loop rotation:48.4°
Quality Score:6.8
Resolution:1.89 Å
Missing Residues:3
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I6
Ligand
No
No
Protein
Yes
Yes

Pocket alignment
Uniprot sequence:EKIGQGASGTVYTVAIKQMLIINEILVMRENKPNIVNYLDSWVVMEYLAGGSLTDVVTEFLHSNQVIHRDIKSDNILLLTDFGFC
Sequence structure:EKIGQGASGTVYTVAIRQMLIINEILVMRENKPNIVNYLDSWVVMEYLAGGSLTDVVTEFLHSNQVIHRNIKSDNILLLTDF___