V-akt murine thymoma viral oncogene homolog 1
Kinase structure
Kinase:AKT1
Family:Akt
Group:AGC
Species:HUMAN
IUPHAR/BPS ID:1479
PDB:4EJN
sc-PDB:
KIDFamMap:Search
Release date:2012-05-23
PubMed: 22533986
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:out
αC-helix conformation:na
G-rich loop angle (distance):65.3° (19Å)
G-rich loop rotation:56.2°
Quality Score:4.4
Resolution:2.19 Å
Missing Residues:7
Missing Atoms:22
Ligand binding mode
Waters
Cluster
I3
I7
Ligand
No
No
Protein
No
No

Allosteric Ligand
Allosteric ligand:0R4
2D structure of the allostericligand
Pocket alignment
Uniprot sequence:KLLGKGTFGKVILYAMKILHTLTENRVLQNSRPFLTALKYSCFVMEYANGGELFFHLSRLHSEKNVVYRDLKLENLMLITDFGLC
Sequence structure:KLLGKGTFGKVILYAMKIL_______VLQNSRPFLTALKYSCFVMEYANGGELFFHLSRLHSEKNVVYRDLKLENLMLITDFGLC