V-akt murine thymoma viral oncogene homolog 1
Kinase structure
Kinase:AKT1
Family:Akt
Group:AGC
Species:HUMAN
IUPHAR/BPS ID:1479
PDB:3O96
sc-PDB:
KIDFamMap:Search
Release date:2010-10-13
PubMed: 20886116
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:out
αC-helix conformation:na
G-rich loop angle (distance):62.6° (19.1Å)
G-rich loop rotation:53.2°
Quality Score:5.2
Resolution:2.7 Å
Missing Residues:5
Missing Atoms:0

Allosteric Ligand
Allosteric ligand:IQO
2D structure of the allostericligand
Pocket alignment
Uniprot sequence:KLLGKGTFGKVILYAMKILHTLTENRVLQNSRPFLTALKYSCFVMEYANGGELFFHLSRLHSEKNVVYRDLKLENLMLITDFGLC
Sequence structure:KLLGKGTFGKVILYAMKIL_____NRVLQNSRPFLTALKYSCFVMEYANGGELFFHLSRLHSEKNVVYRDLKLENLMLITDFGLC