Fibroblast growth factor receptor 1
Kinase structure
Kinase:FGFR1
Family:FGFR
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1808
PDB:4RWI
sc-PDB:
KIDFamMap:Search
Release date:2015-04-15
PubMed: 25686244
Chain:A
(Alternate) Model:A
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The orthosteric binding pocket


More entries for 4RWI
4RWIAlternative model: AChain: B
4RWIAlternative model: BChain: A
4RWIAlternative model: BChain: B


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):62.7° (18.5Å)
G-rich loop rotation:50.6°
Quality Score:8.6
Resolution:2.29 Å
Missing Residues:0
Missing Atoms:14
Ligand binding mode
Waters
Cluster
I4
I5
I6
I11
Ligand
No
No
No
No
Protein
Yes
Yes
No
Yes

Pocket alignment
Uniprot sequence:KPLGEGCFGQVVLVAVKMLDLISEMEMMKMIGKNIINLLGAYVIVEYASKGNLREYLQAYLASKKCIHRDLAARNVLVIADFGLA
Sequence structure:KPLGEGAFGQVVLVAVKMLDLISEMEMMKMIGKNIINLLGAYVIMEYASKGNLREYLQAYLASKKCIHRDLAARNVLVIADFGLA