Search results (215 entries covering 60 PDB structures)

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#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganism DetailsFile
FGFR1FGFRTK7wclAB11-[2,6-bis(fluoranyl)-3,5-dimethoxy-phenyl]-13-ethyl-4-(morpholin-4-ylmethyl)-5,7,11,13-tetrazatricyclo[7.4.0.0^{2,6}]trideca-1(9),2(6),3,7-tetraen-12-oneHumanShow
FGFR1FGFRTK6itjBB4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHumanShow
FGFR1FGFRTK5flfBA-HumanShow
FGFR1FGFRTK5vndAAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHumanShow
FGFR1FGFRTK5ew8BB~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHumanShow
FGFR1FGFRTK5a46BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK3c4fBB3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHumanShow
FGFR1FGFRTK4uwcAB3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHumanShow
FGFR1FGFRTK5uq0AB2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHumanShow
FGFR1FGFRTK2fgiB1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-ureaHumanShow
FGFR1FGFRTK3gqlB(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHumanShow
FGFR1FGFRTK5ur1BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK1fgkBB-HumanShow
FGFR1FGFRTK5am7AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK5flfDA-HumanShow
FGFR1FGFRTK6nvlABn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHumanShow
FGFR1FGFRTK3gqlA(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHumanShow
FGFR1FGFRTK6c19BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK6c1bAB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK6p69ABn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHumanShow
FGFR1FGFRTK6nvlCAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHumanShow
FGFR1FGFRTK4wunABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4nksBAn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK3kxxD-HumanShow
FGFR1FGFRTK5o4aBB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHumanShow
FGFR1FGFRTK5uq0AA2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHumanShow
FGFR1FGFRTK4rwlB6-({7-[(1-aminocyclopropyl)methoxy]-6-methoxyquinolin-4-yl}oxy)-n-methylnaphthalene-1-carboxamideHumanShow
FGFR1FGFRTK6mzwBA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHumanShow
FGFR1FGFRTK3rhxB(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHumanShow
FGFR1FGFRTK4zsaAA4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHumanShow
FGFR1FGFRTK6nvlAAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHumanShow
FGFR1FGFRTK5b7vB[5-amino-1-(2-methyl-1h-benzimidazol-6-yl)-1h-pyrazol-4-yl](1h-indol-2-yl)methanoneHumanShow
FGFR1FGFRTK7ozfABn-[6-(3-ethoxyphenyl)-1h-indazol-3-yl]benzamideHumanShow
FGFR1FGFRTK6c1bBB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK4v05BBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4v01AA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHumanShow
FGFR1FGFRTK5am7BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK5flfBB-HumanShow
FGFR1FGFRTK6p68An-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHumanShow
FGFR1FGFRTK5flfEA-HumanShow
FGFR1FGFRTK4rwkAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK5am6BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK6mzqAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHumanShow
FGFR1FGFRTK3js2B5-(2-thienyl)nicotinic acidHumanShow
FGFR1FGFRTK5o49BB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHumanShow
FGFR1FGFRTK6p68Cn-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHumanShow
FGFR1FGFRTK4rwkBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK5ew8BA~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHumanShow
FGFR1FGFRTK5am6AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK4rwjBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4v05ABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK5z0sBB1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHumanShow
FGFR1FGFRTK3tt0BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHumanShow
FGFR1FGFRTK4f65AA5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4nk9An~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK5flfAA-HumanShow
FGFR1FGFRTK3kxxB-HumanShow
FGFR1FGFRTK5o4aBA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHumanShow
FGFR1FGFRTK4uwbABn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHumanShow
FGFR1FGFRTK1fgkAA-HumanShow
FGFR1FGFRTK6nvlBBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHumanShow
FGFR1FGFRTK6mzqBA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHumanShow
FGFR1FGFRTK6c19BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK5a4cAB1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHumanShow
FGFR1FGFRTK6c1oBAn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHumanShow
FGFR1FGFRTK1fgiBA3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHumanShow
FGFR1FGFRTK6c1cBB7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK6c18BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK1agwBB3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHumanShow
FGFR1FGFRTK5vndBAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHumanShow
FGFR1FGFRTK7ozdAAn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamideHumanShow
FGFR1FGFRTK6c1cAA7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK5ew8AA~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHumanShow
FGFR1FGFRTK4f64BB5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK5zv2A4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamideHumanShow
FGFR1FGFRTK5o49AB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHumanShow
FGFR1FGFRTK4f63B5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK3tt0AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHumanShow
FGFR1FGFRTK5o49BA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHumanShow
FGFR1FGFRTK4wunBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK1fgiAB3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHumanShow
FGFR1FGFRTK4f64AA5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK6c1oBBn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHumanShow
FGFR1FGFRTK5vndBBn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHumanShow
FGFR1FGFRTK4uwbBAn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHumanShow
FGFR1FGFRTK4f63A5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK3js2A5-(2-thienyl)nicotinic acidHumanShow
FGFR1FGFRTK1agwAB3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHumanShow
FGFR1FGFRTK4v01AB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHumanShow
FGFR1FGFRTK6mzwAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHumanShow
FGFR1FGFRTK5am7AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK6mzqBB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHumanShow
FGFR1FGFRTK6nvlDBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHumanShow
FGFR1FGFRTK6p69BAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHumanShow
FGFR1FGFRTK5zv2B4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamideHumanShow
FGFR1FGFRTK4v04AA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHumanShow
FGFR1FGFRTK4uwyAB-HumanShow
FGFR1FGFRTK5a46BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK1fgkAB-HumanShow
FGFR1FGFRTK4v04AB-HumanShow
FGFR1FGFRTK4uwyAA-HumanShow
FGFR1FGFRTK6nvlCBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHumanShow
FGFR1FGFRTK3ky2B-HumanShow
FGFR1FGFRTK6p68Bn-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHumanShow
FGFR1FGFRTK4rwjABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK5flfEB-HumanShow
FGFR1FGFRTK3c4fBA3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHumanShow
FGFR1FGFRTK4rwjAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4f65BA5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK1fgkBA-HumanShow
FGFR1FGFRTK6c18AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK1agwAA3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHumanShow
FGFR1FGFRTK5a4cAA1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHumanShow
FGFR1FGFRTK4nk9Bn~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK7ozbAB4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHumanShow
FGFR1FGFRTK5ur1BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK4uwyBA-HumanShow
FGFR1FGFRTK4f64BA5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4rwkABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK1fgiAA3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHumanShow
FGFR1FGFRTK3c4fAA3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHumanShow
FGFR1FGFRTK5uq0BA2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHumanShow
FGFR1FGFRTK8jmzAAn-(2-(dimethylamino)ethyl)-1-(3-((4-((2-methyl-1h-indol-5-yl)oxy)pyrimidin-2-yl)amino)phenyl)methanesulfonamideHumanShow
FGFR1FGFRTK6c1bBA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK4rwkBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4zsaAB4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHumanShow
FGFR1FGFRTK4v01BA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHumanShow
FGFR1FGFRTK4uwbBBn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHumanShow
FGFR1FGFRTK3tt0AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHumanShow
FGFR1FGFRTK4nksAAn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK6c19AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK3ky2A-HumanShow
FGFR1FGFRTK5am6BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK5o4aAA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHumanShow
FGFR1FGFRTK4rwiBB-HumanShow
FGFR1FGFRTK5flfCB-HumanShow
FGFR1FGFRTK5a4cBB1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHumanShow
FGFR1FGFRTK5o4aAB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHumanShow
FGFR1FGFRTK6c1oAAn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHumanShow
FGFR1FGFRTK5b7vA[5-amino-1-(2-methyl-1h-benzimidazol-6-yl)-1h-pyrazol-4-yl](1h-indol-2-yl)methanoneHumanShow
FGFR1FGFRTK4nksBBn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4uwcBA3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHumanShow
FGFR1FGFRTK4rwjBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4zsaBA4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHumanShow
FGFR1FGFRTK3kxxA-HumanShow
FGFR1FGFRTK4v04BB-HumanShow
FGFR1FGFRTK1agwBA3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHumanShow
FGFR1FGFRTK4nksABn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK5a4cBA1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHumanShow
FGFR1FGFRTK5vndABn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHumanShow
FGFR1FGFRTK4nkaAn~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4zsaBB4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHumanShow
FGFR1FGFRTK6mzwAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHumanShow
FGFR1FGFRTK6mzqAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHumanShow
FGFR1FGFRTK8jmzABn-(2-(dimethylamino)ethyl)-1-(3-((4-((2-methyl-1h-indol-5-yl)oxy)pyrimidin-2-yl)amino)phenyl)methanesulfonamideHumanShow
FGFR1FGFRTK5z0sAA1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHumanShow
FGFR1FGFRTK6itjBA4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHumanShow
FGFR1FGFRTK6c18BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK4f64AB5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4uwcAA3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHumanShow
FGFR1FGFRTK3tt0BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHumanShow
FGFR1FGFRTK4rwlA-HumanShow
FGFR1FGFRTK3c4fAB3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHumanShow
FGFR1FGFRTK5flfAB-HumanShow
FGFR1FGFRTK5z0sAB1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHumanShow
FGFR1FGFRTK4nkaBn~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4uwbAAn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHumanShow
FGFR1FGFRTK5a46AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK6c1oABn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHumanShow
FGFR1FGFRTK3kxxC-HumanShow
FGFR1FGFRTK2fgiA1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-ureaHumanShow
FGFR1FGFRTK7ozdABn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamideHumanShow
FGFR1FGFRTK3gqlC(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHumanShow
FGFR1FGFRTK5ur1AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK1fgiBB3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHumanShow
FGFR1FGFRTK5am6AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK6mzwBB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHumanShow
FGFR1FGFRTK5am7BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK6itjAA4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHumanShow
FGFR1FGFRTK6c19AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK5flfCA-HumanShow
FGFR1FGFRTK6nvlBAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHumanShow
FGFR1FGFRTK7ozbAA4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHumanShow
FGFR1FGFRTK5ur1AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK6c1bAA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK4rwiAA-HumanShow
FGFR1FGFRTK6c1cBA7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK6p69AAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHumanShow
FGFR1FGFRTK6p69BBn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHumanShow
FGFR1FGFRTK4v04BA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHumanShow
FGFR1FGFRTK4v05AAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK4uwyBB-HumanShow
FGFR1FGFRTK5uq0BB2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHumanShow
FGFR1FGFRTK4uwcBB3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHumanShow
FGFR1FGFRTK6c18AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK4v01BB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHumanShow
FGFR1FGFRTK4f65BB5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK7wclAA11-[2,6-bis(fluoranyl)-3,5-dimethoxy-phenyl]-13-ethyl-4-(morpholin-4-ylmethyl)-5,7,11,13-tetrazatricyclo[7.4.0.0^{2,6}]trideca-1(9),2(6),3,7-tetraen-12-oneHumanShow
FGFR1FGFRTK5a46AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHumanShow
FGFR1FGFRTK6c1cAB7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHumanShow
FGFR1FGFRTK4wunAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK3gqiAphosphomethylphosphonic acid adenylate esterHumanShow
FGFR1FGFRTK4v05BAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow
FGFR1FGFRTK7ozfAAn-[6-(3-ethoxyphenyl)-1h-indazol-3-yl]benzamideHumanShow
FGFR1FGFRTK4rwiAB-HumanShow
FGFR1FGFRTK5z0sBA1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHumanShow
FGFR1FGFRTK5o49AA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHumanShow
FGFR1FGFRTK6itjAB4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHumanShow
FGFR1FGFRTK6nvlDAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHumanShow
FGFR1FGFRTK3rhxA(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHumanShow
FGFR1FGFRTK5ew8AB~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHumanShow
FGFR1FGFRTK4rwiBA-HumanShow
FGFR1FGFRTK5flfDB-HumanShow
FGFR1FGFRTK4f65AB5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHumanShow
FGFR1FGFRTK4wunBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHumanShow