Fibroblast growth factor receptor 1
Kinase structure
Kinase:FGFR1
Family:FGFR
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1808
PDB:4RWI
sc-PDB:
KIDFamMap:Search
Release date:2015-04-15
PubMed: 25686244
Chain:B
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 4RWI
4RWIAlternative model: AChain: A
4RWIAlternative model: AChain: B
4RWIAlternative model: BChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):63° (18.7Å)
G-rich loop rotation:42.7°
Quality Score:8.8
Resolution:2.29 Å
Missing Residues:2
Missing Atoms:4
Ligand binding mode
Waters
Cluster
I4
Ligand
No
Protein
Yes

Pocket alignment
Uniprot sequence:KPLGEGCFGQVVLVAVKMLDLISEMEMMKMIGKNIINLLGAYVIVEYASKGNLREYLQAYLASKKCIHRDLAARNVLVIADFGLA
Sequence structure:KPLGEG__GQVVLVAVKMLDLISEMEMMKMIGKNIINLLGAYVIMEYASKGNLREYLQAYLASKKCIHRDLAARNVLVIADFGLA