Cyclin-dependent kinase 8
Kinase structure
Kinase:CDK8
Family:CDK
Group:CMGC
Species:HUMAN
IUPHAR/BPS ID:1980
PDB:4G6L
sc-PDB:
KIDFamMap:Search
Release date:2013-05-01
PubMed: 23630251
Chain:A
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The orthosteric binding pocket
Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):52.7° (16.2Å)
G-rich loop rotation:46.1°
Quality Score:8
Resolution:2.7 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I5
Ligand
No
Protein
Yes

Pocket alignment
Uniprot sequence:CKVGRGTYGHVYKYALKQISACREIALLRELKPNVISLQKVWLLFDYAE-HDLWHIIKFYLHANWVLHRDLKPANILVIADMGFA
Sequence structure:CKVGRGTYGHVYKYALKQISACREIALLRELKPNVISLQKVWLLFDYAE_HDLWHIIKFYLHANWVLHRDLKPANILVIADMGFA