Mitogen-activated protein kinase 14
Kinase structure
Kinase:MAPK14 (p38a)
Family:MAPK
Group:CMGC
Species:HUMAN
IUPHAR/BPS ID:1499
PDB:4E8A
sc-PDB:
KIDFamMap:Search
Release date:2012-10-31
PubMed: 23079240
Chain:A
Click to open a 3D viewer
The orthosteric binding pocket
Structural information
DFG conformation:na
αC-helix conformation:in
G-rich loop angle (distance):68.9° (20.2Å)
G-rich loop rotation:22.5°
Quality Score:4
Resolution:2.7 Å
Missing Residues:9
Missing Atoms:0

Allosteric Ligand
Allosteric ligand:0OA
2D structure of the allostericligand
Pocket alignment
Uniprot sequence:SPVGSGAYGSVCAVAVKKLRTYRELRLLKHMKENVIGLLDVYLVTHLMG-ADLNNIVKCYIHSADIIHRDLKPSNLAVILDFGLA
Sequence structure:SPVG_GAYGSVCAVAVKKLRTYRELRLLKHMKENVIGLLDVYLVTHLMG_ADLNN____YIHSADIIHRDLKPSNLAVILD____