Insulin receptor
Kinase structure
Kinase:INSR
Family:InsR
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1800
PDB:2B4S
sc-PDB:
KIDFamMap:Search
Release date:2005-11-15
PubMed: 16271887
Chain:D
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The orthosteric binding pocket


More entries for 2B4S
2B4SChain: B


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):50.3° (15.1Å)
G-rich loop rotation:81.9°
Quality Score:8
Resolution:2.3 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I8
Ligand
No
Protein
No

Pocket alignment
Uniprot sequence:RELGQGSFGMVYEVAVKTVEFLNEASVMKGFT-HVVRLLGVLVVMELMAHGDLKSYLRSYLNAKKFVHRDLAARNCMVIGDFGMT
Sequence structure:RELGQGSFGMVYEVAVKTVEFLNEASVMKGFT_HVVRLLGVLVVMELMAHGDLKSYLRSYLNAKKFVHRDLAARNCMVIGDFGMT