Insulin receptor
Kinase structure
Kinase:INSR
Family:InsR
Group:TK
Species:HUMAN
IUPHAR/BPS ID:1800
PDB:1IRK
sc-PDB:
KIDFamMap:Search
Release date:1995-02-27
PubMed: 7997262
Chain:A
(Alternate) Model:A
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The orthosteric binding pocket


More entries for 1IRK
1IRKAlternative model: BChain: A


Structural information
DFG conformation:out
αC-helix conformation:out
G-rich loop angle (distance):65.7° (18.8Å)
G-rich loop rotation:74.4°
Quality Score:7.2
Resolution:2.1 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I6
Ligand
No
No
Protein
Yes
Yes

Pocket alignment
Uniprot sequence:RELGQGSFGMVYEVAVKTVEFLNEASVMKGFT-HVVRLLGVLVVMELMAHGDLKSYLRSYLNAKKFVHRDLAARNCMVIGDFGMT
Sequence structure:RELGQGSFGMVYEVAVKTVEFLNEASVMKGFT_HVVRLLGVLVVMELMAHGDLKSYLRSYLNAKKFVHRDLAARNCMVIGDFGMT