B-Raf proto-oncogene, serine/threonine kinase
Kinase structure
Kinase:BRAF
Family:RAF
Group:TKL
Species:HUMAN
IUPHAR/BPS ID:1943
PDB:4XV3
sc-PDB:
KIDFamMap:Search
Release date:2015-10-28
PubMed: 26466569
Chain:B
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The orthosteric binding pocket


More entries for 4XV3
4XV3Chain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):-
G-rich loop rotation:-
Quality Score:4.8
Resolution:2.8 Å
Missing Residues:8
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I5
Ligand
No
Protein
Yes

Pocket alignment
Uniprot sequence:QRIGSGSFGTVYKVAVKMLAFKNEVGVLRKTRVNILLFMGYAIVTQWCEGSSLYHHLHIYLHAKSIIHRDLKSNNIFLIGDFGLA
Sequence structure:QRIG______VYKVAVKMLAFKNEVGVLRKTRVNILLFMGYAIVTQWCEGSSLYHHLHAYLHAKSIIHRDLKSNNIFLIGDF__A