Transforming growth factor beta receptor I
Kinase structure
Kinase:TGFBR1 (TGFbR1)
Family:STKR
Group:TKL
Species:HUMAN
IUPHAR/BPS ID:1788
PDB:5E8S
sc-PDB:
KIDFamMap:Search
Release date:2016-05-11
PubMed: 27139629
Chain:A
(Alternate) Model:B
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The orthosteric binding pocket


More entries for 5E8S
5E8SAlternative model: AChain: A


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):54.5° (16.1Å)
G-rich loop rotation:61.7°
Quality Score:9.8
Resolution:1.45 Å
Missing Residues:0
Missing Atoms:2
Ligand binding mode
Waters
Cluster
I1
I2
I5
I8
Ligand
No
No
No
No
Protein
Yes
Yes
Yes
Yes

Pocket alignment
Uniprot sequence:ESIGKGRFGEVWRVAVKIFSWFREAEIYQTVMENILGFIAAWLVSDYHEHGSLFDYLNRTQGKPAIAHRDLKSKNILVIADLGLA
Sequence structure:ESIGKGRFGEVWRVAVKIFSWFREAEIYQTVMENILGFIAAWLVSDYHEHGSLFDYLNRTQGKPAIAHRDLKSKNILVIADLGLA