Endoplasmic reticulum to nucleus signaling 1
Kinase structure
Kinase:ERN1 (IRE1)
Family:IRE
Group:Other
Species:HUMAN
IUPHAR/BPS ID:2020
PDB:5HGI
sc-PDB:
KIDFamMap:Search
Release date:2016-06-08
PubMed: 27227314
Chain:A
Click to open a 3D viewer
The orthosteric binding pocket
Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):-
G-rich loop rotation:-
Quality Score:6.8
Resolution:2.58 Å
Missing Residues:3
Missing Atoms:49
Ligand binding mode
Waters
Cluster
I5
Ligand
No
Protein
Yes

Pocket alignment
Uniprot sequence:DVLGHGAEGTIVYVAVKRIFADREVQLLRESDPNVIRYFCTYIAIELCAA-TLQEYVEQHLHSLNIVHRDLKPHNILIISDFGLC
Sequence structure:DVLGHG___TIVYVAVKRIFADREVQLLRESDPNVIRYFCTYIAIELCAA_TLQEYVEQHLHSLNIVHRDLKPHNILIISDFGLC