Protein kinase cAMP-activated catalytic subunit alpha
Kinase structure
Kinase:PRKACA (PKACa)
Family:PKA
Group:AGC
Species:HUMAN
IUPHAR/BPS ID:1476
PDB:5IZJ
sc-PDB:
KIDFamMap:Search
Release date:2016-07-20
PubMed: 27389935
Chain:A
(Alternate) Model:B
Click to open a 3D viewer
The orthosteric binding pocket


More entries for 5IZJ
5IZJAlternative model: AChain: A
5IZJAlternative model: AChain: B
5IZJAlternative model: BChain: B


Structural information
DFG conformation:in
αC-helix conformation:in
G-rich loop angle (distance):63.2° (19.5Å)
G-rich loop rotation:53.1°
Quality Score:8
Resolution:1.85 Å
Missing Residues:0
Missing Atoms:0
Ligand binding mode
Waters
Cluster
I1
I4
I5
Ligand
No
No
No
Protein
Yes
Yes
Yes

Allosteric Ligand
Allosteric ligand:6J9
2D structure of the allostericligand
Pocket alignment
Uniprot sequence:KTLGTGSFGRVMLYAMKILHTLNEKRILQAVNPFLVKLEFSYMVMEYVPGGEMFSHLRRYLHSLDLIYRDLKPENLLIVTDFGFA
Sequence structure:KTLGTGSFGRVMLYAMKILHTLNEKRILQAVNPFLVKLEFSYMVMEYVPGGEMFSHLRRYLHSLDLIYRDLKPENLLIVTDFGFA